TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois College of Pharmacy
Curated by ChEMBL
University of Illinois College of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 2.40nMAssay Description:Antagonist activity at ERalpha in tamoxifen-sensitive human MCF7:WS8 cells assessed as inhibition of estradiol-induced response after 18 hrs by lucif...More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois College of Pharmacy
Curated by ChEMBL
University of Illinois College of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 3.10nMAssay Description:Antagonist activity at ERalpha in tamoxifen-sensitive human MCF7:WS8 cells assessed as inhibition of estradiol-induced response after 18 hrs by lucif...More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois College of Pharmacy
Curated by ChEMBL
University of Illinois College of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Antagonist activity at ERalpha in tamoxifen-sensitive human MCF7:WS8 cells assessed as inhibition of estradiol-induced response after 18 hrs by lucif...More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois College of Pharmacy
Curated by ChEMBL
University of Illinois College of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:Antagonist activity at ERalpha in tamoxifen-sensitive human MCF7:WS8 cells assessed as inhibition of estradiol-induced response after 18 hrs by lucif...More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois College of Pharmacy
Curated by ChEMBL
University of Illinois College of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 8.80nMAssay Description:Antagonist activity at ERalpha in tamoxifen-sensitive human MCF7:WS8 cells assessed as inhibition of estradiol-induced response after 18 hrs by lucif...More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois College of Pharmacy
Curated by ChEMBL
University of Illinois College of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Antagonist activity at ERalpha in tamoxifen-sensitive human MCF7:WS8 cells assessed as inhibition of estradiol-induced response after 18 hrs by lucif...More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois College of Pharmacy
Curated by ChEMBL
University of Illinois College of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Antagonist activity at ERalpha in tamoxifen-sensitive human MCF7:WS8 cells assessed as inhibition of estradiol-induced response after 18 hrs by lucif...More data for this Ligand-Target Pair
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