Affinity DataIC50: 0.5nMAssay Description:Displacement of [3H]-1,25(OH)2D3 from GST-fused human VDR-LBD expressed in Escherichia coli BL21More data for this Ligand-Target Pair
Affinity DataIC50: 8.5nMAssay Description:Inhibition of CYP2C19More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]-1,25(OH)2D3 from GST-fused human VDR-LBD expressed in Escherichia coli BL21More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]-1,25(OH)2D3 from GST-fused human VDR-LBD expressed in Escherichia coli BL21More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Displacement of [3H]-1,25(OH)2D3 from GST-fused human VDR-LBD expressed in Escherichia coli BL21More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of CYP2C19More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase IMP-1(Pseudomonas aeruginosa)
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 1.55E+3nMAssay Description:Inhibition of carbapenems-resistant Pseudomonas aeruginosa MSC15369 metallo-beta-lactamase IMP1 expressed in Escherichia coli DH5[alpha] using nitroc...More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase IMP-1(Pseudomonas aeruginosa)
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of carbapenems-resistant Pseudomonas aeruginosa MSC15369 metallo-beta-lactamase IMP1 expressed in Escherichia coli DH5[alpha] using nitroc...More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase IMP-1(Pseudomonas aeruginosa)
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of carbapenems-resistant Pseudomonas aeruginosa MSC15369 metallo-beta-lactamase IMP1 expressed in Escherichia coli DH5[alpha] using nitroc...More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase IMP-1(Pseudomonas aeruginosa)
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of carbapenems-resistant Pseudomonas aeruginosa MSC15369 metallo-beta-lactamase IMP1 expressed in Escherichia coli DH5[alpha] using nitroc...More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase IMP-1(Pseudomonas aeruginosa)
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of carbapenems-resistant Pseudomonas aeruginosa MSC15369 metallo-beta-lactamase IMP1 expressed in Escherichia coli DH5[alpha] using nitroc...More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase IMP-1(Pseudomonas aeruginosa)
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of carbapenems-resistant Pseudomonas aeruginosa MSC15369 metallo-beta-lactamase IMP1 expressed in Escherichia coli DH5[alpha] using nitroc...More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase IMP-1(Pseudomonas aeruginosa)
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of carbapenems-resistant Pseudomonas aeruginosa MSC15369 metallo-beta-lactamase IMP1 expressed in Escherichia coli DH5[alpha] using nitroc...More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase IMP-1(Pseudomonas aeruginosa)
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of carbapenems-resistant Pseudomonas aeruginosa MSC15369 metallo-beta-lactamase IMP1 expressed in Escherichia coli DH5[alpha] using nitroc...More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase IMP-1(Pseudomonas aeruginosa)
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of carbapenems-resistant Pseudomonas aeruginosa MSC15369 metallo-beta-lactamase IMP1 expressed in Escherichia coli DH5[alpha] using nitroc...More data for this Ligand-Target Pair
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase IMP-1(Pseudomonas aeruginosa)
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of carbapenems-resistant Pseudomonas aeruginosa MSC15369 metallo-beta-lactamase IMP1 expressed in Escherichia coli DH5[alpha] using nitroc...More data for this Ligand-Target Pair
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of CYP1A2More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase IMP-1(Pseudomonas aeruginosa)
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of carbapenems-resistant Pseudomonas aeruginosa MSC15369 metallo-beta-lactamase IMP1 expressed in Escherichia coli DH5[alpha] using nitroc...More data for this Ligand-Target Pair
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase IMP-1(Pseudomonas aeruginosa)
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of carbapenems-resistant Pseudomonas aeruginosa MSC15369 metallo-beta-lactamase IMP1 expressed in Escherichia coli DH5[alpha] using nitroc...More data for this Ligand-Target Pair
Affinity DataIC50: 8.60E+3nMAssay Description:Inhibition of CYP1A2More data for this Ligand-Target Pair
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase IMP-1(Pseudomonas aeruginosa)
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibition of carbapenems-resistant Pseudomonas aeruginosa MSC15369 metallo-beta-lactamase IMP1 expressed in Escherichia coli DH5[alpha] using nitroc...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of CYP2C19More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase IMP-1(Pseudomonas aeruginosa)
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 1.31E+4nMAssay Description:Inhibition of carbapenems-resistant Pseudomonas aeruginosa MSC15369 metallo-beta-lactamase IMP1 expressed in Escherichia coli DH5[alpha] using nitroc...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase IMP-1(Pseudomonas aeruginosa)
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 1.88E+4nMAssay Description:Inhibition of carbapenems-resistant Pseudomonas aeruginosa MSC15369 metallo-beta-lactamase IMP1 expressed in Escherichia coli DH5[alpha] using nitroc...More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase IMP-1(Pseudomonas aeruginosa)
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 2.14E+4nMAssay Description:Inhibition of carbapenems-resistant Pseudomonas aeruginosa MSC15369 metallo-beta-lactamase IMP1 expressed in Escherichia coli DH5[alpha] using nitroc...More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase IMP-1(Pseudomonas aeruginosa)
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 2.56E+4nMAssay Description:Inhibition of carbapenems-resistant Pseudomonas aeruginosa MSC15369 metallo-beta-lactamase IMP1 expressed in Escherichia coli DH5[alpha] using nitroc...More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase IMP-1(Pseudomonas aeruginosa)
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 4.78E+4nMAssay Description:Inhibition of carbapenems-resistant Pseudomonas aeruginosa MSC15369 metallo-beta-lactamase IMP1 expressed in Escherichia coli DH5[alpha] using nitroc...More data for this Ligand-Target Pair
Affinity DataIC50: 9.40E+4nMAssay Description:Inhibition of CYP1A2More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase IMP-1(Pseudomonas aeruginosa)
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 9.45E+4nMAssay Description:Inhibition of carbapenems-resistant Pseudomonas aeruginosa MSC15369 metallo-beta-lactamase IMP1 expressed in Escherichia coli DH5[alpha] using nitroc...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of CYP1A2More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase IMP-1(Pseudomonas aeruginosa)
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 1.42E+5nMAssay Description:Inhibition of carbapenems-resistant Pseudomonas aeruginosa MSC15369 metallo-beta-lactamase IMP1 expressed in Escherichia coli DH5[alpha] using nitroc...More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase IMP-1(Pseudomonas aeruginosa)
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of carbapenems-resistant Pseudomonas aeruginosa MSC15369 metallo-beta-lactamase IMP1 expressed in Escherichia coli DH5[alpha] using nitroc...More data for this Ligand-Target Pair
TargetMetallo-beta-lactamase IMP-1(Pseudomonas aeruginosa)
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Meiji Seika Pharma, Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of carbapenems-resistant Pseudomonas aeruginosa MSC15369 metallo-beta-lactamase IMP1 expressed in Escherichia coli DH5[alpha] using nitroc...More data for this Ligand-Target Pair
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