Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1A adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 0.794nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.930nMAssay Description:Binding affinity against alpha-2 adrenergic receptor from calf cerebral cortex, using [3H]prazosin as the radioligandMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Compound was evaluated for binding affinity towards dopamine receptor D2 in striatal membranes, using [3H]- spiperone as radioligand in the presence ...More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
UnWersity of Misscuri
Curated by PDSP Ki Database
UnWersity of Misscuri
Curated by PDSP Ki Database
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Institut de Recherches Servier, Centre de Recherches de Croissy
Curated by PDSP Ki Database
Institut de Recherches Servier, Centre de Recherches de Croissy
Curated by PDSP Ki Database
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Institut de Recherches Servier, Centre de Recherches de Croissy
Curated by PDSP Ki Database
Institut de Recherches Servier, Centre de Recherches de Croissy
Curated by PDSP Ki Database
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]RX781094 from alpha2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Binding affinity against alpha-2 adrenergic receptor from calf cerebral cortex, using [3H]prazosin as the radioligandMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Institut de Recherches Servier, Centre de Recherches de Croissy
Curated by PDSP Ki Database
Institut de Recherches Servier, Centre de Recherches de Croissy
Curated by PDSP Ki Database
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Institut de Recherches Servier, Centre de Recherches de Croissy
Curated by PDSP Ki Database
Institut de Recherches Servier, Centre de Recherches de Croissy
Curated by PDSP Ki Database
Affinity DataKi: 2.60nMAssay Description:The compound was tested for binding affinity against Alpha-2A adrenergic receptor from human clones.More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
UnWersity of Misscuri
Curated by PDSP Ki Database
UnWersity of Misscuri
Curated by PDSP Ki Database
TargetAlpha-2A adrenergic receptor [16-465](Rattus norvegicus (rat))
Glaxo SmithKline Pharmaceuticals
Curated by PDSP Ki Database
Glaxo SmithKline Pharmaceuticals
Curated by PDSP Ki Database
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Institut de Recherches Servier, Centre de Recherches de Croissy
Curated by PDSP Ki Database
Institut de Recherches Servier, Centre de Recherches de Croissy
Curated by PDSP Ki Database
Affinity DataKi: 4.10nMAssay Description:Binding affinity towards alpha-1A adrenergic receptor expressed in human embryonic kidney (HEK293) cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
UnWersity of Misscuri
Curated by PDSP Ki Database
UnWersity of Misscuri
Curated by PDSP Ki Database
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Institut de Recherches Servier, Centre de Recherches de Croissy
Curated by PDSP Ki Database
Institut de Recherches Servier, Centre de Recherches de Croissy
Curated by PDSP Ki Database
TargetAlpha-2A adrenergic receptor [16-465](Rattus norvegicus (rat))
Glaxo SmithKline Pharmaceuticals
Curated by PDSP Ki Database
Glaxo SmithKline Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 4.70nMAssay Description:The compound was tested for binding affinity against alpha-2D adrenergic receptor, from rat clones.More data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1B adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465](Rattus norvegicus (rat))
Glaxo SmithKline Pharmaceuticals
Curated by PDSP Ki Database
Glaxo SmithKline Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 5nMAssay Description:Binding affinity against alpha-2-adrenergic receptor using 10 nM [3H]yohimbine in human platelet membranes from three separate experiments using 10 i...More data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Institut de Recherches Servier, Centre de Recherches de Croissy
Curated by PDSP Ki Database
Institut de Recherches Servier, Centre de Recherches de Croissy
Curated by PDSP Ki Database
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Institut de Recherches Servier, Centre de Recherches de Croissy
Curated by PDSP Ki Database
Institut de Recherches Servier, Centre de Recherches de Croissy
Curated by PDSP Ki Database
TargetAlpha-2A adrenergic receptor [16-465](Rattus norvegicus (rat))
Glaxo SmithKline Pharmaceuticals
Curated by PDSP Ki Database
Glaxo SmithKline Pharmaceuticals
Curated by PDSP Ki Database
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University of Nebraska
Curated by PDSP Ki Database
University of Nebraska
Curated by PDSP Ki Database
Affinity DataKi: 6.80nMAssay Description:Displacement of [3H]prazosin (0.3 nM) from bovine Alpha-1A adrenergic receptor expressed in BHK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.60nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1D adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University of Nebraska
Curated by PDSP Ki Database
University of Nebraska
Curated by PDSP Ki Database
Affinity DataKi: 7.60nMAssay Description:Binding affinity against Alpha-2B adrenergic receptor from human clones.More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
UnWersity of Misscuri
Curated by PDSP Ki Database
UnWersity of Misscuri
Curated by PDSP Ki Database
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Institut de Recherches Servier, Centre de Recherches de Croissy
Curated by PDSP Ki Database
Institut de Recherches Servier, Centre de Recherches de Croissy
Curated by PDSP Ki Database
Affinity DataKi: 8.40nMAssay Description:Binding affinity against Alpha-2C adrenergic receptor from human clones.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataKi: 9.30nMAssay Description:Compound was tested for the inhibition of [3H]clonidine binding Alpha-2 adrenergic receptor of crude rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 9.80nMAssay Description:Compound was tested for the inhibition of [3H]prazosin binding Alpha-1 adrenergic receptor of crude rat brain membrane.More data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University of Nebraska
Curated by PDSP Ki Database
University of Nebraska
Curated by PDSP Ki Database
Affinity DataKi: 10nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenoceptor in rat cerebral cortex after 30 mins by beta scintillation countingMore data for this Ligand-Target Pair