Compile Data Set for Download or QSAR
Found 41 of ki for monomerid = 50381677
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]U-69593 from human recombinant Opioid receptor kappa 1 on CHO cell membranes.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27945F9PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cell membranes incubated for 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X58ZXPubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  0.700nMAssay Description:Displacement of radiolabeled U69593 from kappa1 opioid receptor in Hartley guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XG9RXFPubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  0.880nMAssay Description:Displacement of [3H]U-69593 from kappa-opoid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2X2RPubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  0.970nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain membranes after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G73GDPPubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  0.970nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig brain membrane after 150 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ59RZPubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor transfected in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5QC2PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Binding affinity against opioid receptor kappa 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M08QQPubMed
TargetMu-type opioid receptor(MOUSE)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Binding affinity against opioid receptor by displacing radioligand [3HlU69,593More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M32WD4PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MPCPubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]U-69593 from guinea pig cerebellum KORMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53NFKPubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]U69593 from human KOP receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0V9TPubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Binding affinity determined against Opioid receptor kappa 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M08QQPubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]-U69593 from human kappa opioid receptor expressed in CHO cells membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC03ZQPubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]U69,593 from human recombinant opioid kappa receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0W6WPubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  4.80nMAssay Description:Binding affinity at Opioid receptor kappa 1 by displacement of [3H]U-69593 in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2639QGWPubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Universit£ di Chieti-Pescara"G. d'Annunzio"

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in Wistar rat brain membranes by liquid scintillation counting based competition binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9JS5PubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  391nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain membranes without cerebellum after 1 hr by liquid scintillation counting an...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MPCPubMed
TargetMu-type opioid receptor(MOUSE)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  548nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain membranes without cerebellum after 1 hr by liquid scintillation counting analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348MPCPubMed
TargetMu-type opioid receptor(GUINEA PIG)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  692nMAssay Description:Displacement of radiolabeled DAMGO from mu opioid receptor in Hartley guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XG9RXFPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity determined against Opioid receptor mu 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M08QQPubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DPDPE from mouse whole brain DORMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53NFKPubMed
TargetMu-type opioid receptor(MOUSE)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mouse whole brain MORMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53NFKPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity determined against Opioid receptor delta 1 from human cloned receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M08QQPubMed
TargetNociceptin receptor(Cavia porcellus)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of radiolabeled NalBzOH from kappa3 opioid receptor in Hartley guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XG9RXFPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  1.15E+3nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cell membranes incubated for 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X58ZXPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  1.15E+3nMAssay Description:Displacement of [3H]DAMGO from human recombinant Opioid receptor mu 1 on CHO cell membranes.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27945F9PubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  1.36E+3nMAssay Description:Displacement of radiolabeled DPDPE-Cl from delta opioid receptor in Hartley guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XG9RXFPubMed
TargetMu-type opioid receptor(GUINEA PIG)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  1.88E+3nMAssay Description:Binding affinity of compound was determined against Opioid receptor mu 1 from native receptor in guinea pigMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M08QQPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [3H]DAMGO from human recombinant opioid mu receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting meth...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0W6WPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  2.37E+3nMAssay Description:Displacement of [3H]-DAMGO from human mu opioid receptor expressed in CHO cells membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC03ZQPubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity at opioid receptor delta 1 by displacement of [3H]DADLE in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2639QGWPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Southern Research Institute

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  7.25E+3nMAssay Description:Binding affinity at Opioid receptor mu 1 by displacement of [3H]DAMGO in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2639QGWPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]pCl-DPDPE from human delta opioid receptor expressed in CHO cell membranes incubated for 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X58ZXPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]C1-DPDPE from human recombinant Opioid receptor delta 1 on CHO cell membranes.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27945F9PubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Cl-DPDPE from human DOP receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0V9TPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DAMGO from human MOP receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0V9TPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity of compound was determined against Opioid receptor delta 1 from a native receptor in guinea pigMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M08QQPubMed
TargetNociceptin receptor(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Partial agonist activity at human NOP receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding after 60 mins by scintillatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0V9TPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi: >1.20E+4nMAssay Description:Displacement of [3H]DADLE from human recombinant opioid delta receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0W6WPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  1.25E+4nMAssay Description:Displacement of [3H]-DADLE from human delta opioid receptor expressed in CHO cells membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC03ZQPubMed