TargetBile acid receptor(Homo sapiens (Human))
Institute of Pharmaceutical Chemistry, Goethe-University Frankfurt , Max-von-Laue-Strasse 9, D-60438 Frankfurt am Main, Germany.
Curated by ChEMBL
Institute of Pharmaceutical Chemistry, Goethe-University Frankfurt , Max-von-Laue-Strasse 9, D-60438 Frankfurt am Main, Germany.
Curated by ChEMBL
Affinity DataKd: 37nMAssay Description:Binding affinity to FXR (unknown origin) ligand binding domain by ITC assayMore data for this Ligand-Target Pair
TargetBile acid receptor(Homo sapiens (Human))
Institute of Pharmaceutical Chemistry, Goethe-University Frankfurt , Max-von-Laue-Strasse 9, D-60438 Frankfurt am Main, Germany.
Curated by ChEMBL
Institute of Pharmaceutical Chemistry, Goethe-University Frankfurt , Max-von-Laue-Strasse 9, D-60438 Frankfurt am Main, Germany.
Curated by ChEMBL
Affinity DataKd: 130nMAssay Description:Binding affinity to FXR ligand binding domain (unknown origin) isothermal titration calorimetry assayMore data for this Ligand-Target Pair
TargetBile acid receptor(Homo sapiens (Human))
Institute of Pharmaceutical Chemistry, Goethe-University Frankfurt , Max-von-Laue-Strasse 9, D-60438 Frankfurt am Main, Germany.
Curated by ChEMBL
Institute of Pharmaceutical Chemistry, Goethe-University Frankfurt , Max-von-Laue-Strasse 9, D-60438 Frankfurt am Main, Germany.
Curated by ChEMBL
Affinity DataKd: 300nMAssay Description:Binding affinity to recombinant FXR-LBD (unknown origin) expressed in Escherichia coli BL21 (DE3) gold cells by isothermal titration calorimetryMore data for this Ligand-Target Pair
TargetBile acid receptor(Homo sapiens (Human))
Institute of Pharmaceutical Chemistry, Goethe-University Frankfurt , Max-von-Laue-Strasse 9, D-60438 Frankfurt am Main, Germany.
Curated by ChEMBL
Institute of Pharmaceutical Chemistry, Goethe-University Frankfurt , Max-von-Laue-Strasse 9, D-60438 Frankfurt am Main, Germany.
Curated by ChEMBL
Affinity DataKd: 4.00E+3nMAssay Description:Binding affinity to recombinant FXR-LBD (unknown origin) expressed in Escherichia coli BL21 (DE3) gold cells by isothermal titration calorimetryMore data for this Ligand-Target Pair
TargetBile acid receptor(Homo sapiens (Human))
Institute of Pharmaceutical Chemistry, Goethe-University Frankfurt , Max-von-Laue-Strasse 9, D-60438 Frankfurt am Main, Germany.
Curated by ChEMBL
Institute of Pharmaceutical Chemistry, Goethe-University Frankfurt , Max-von-Laue-Strasse 9, D-60438 Frankfurt am Main, Germany.
Curated by ChEMBL
Affinity DataKd: 9.00E+3nMAssay Description:Binding affinity to recombinant FXR-LBD (unknown origin) expressed in Escherichia coli BL21 (DE3) gold cells by isothermal titration calorimetryMore data for this Ligand-Target Pair
TargetBile acid receptor(Homo sapiens (Human))
Institute of Pharmaceutical Chemistry, Goethe-University Frankfurt , Max-von-Laue-Strasse 9, D-60438 Frankfurt am Main, Germany.
Curated by ChEMBL
Institute of Pharmaceutical Chemistry, Goethe-University Frankfurt , Max-von-Laue-Strasse 9, D-60438 Frankfurt am Main, Germany.
Curated by ChEMBL
Affinity DataKd: 4.87E+4nMAssay Description:Binding affinity to FXR (unknown origin)More data for this Ligand-Target Pair
TargetBile acid receptor(Homo sapiens (Human))
Institute of Pharmaceutical Chemistry, Goethe-University Frankfurt , Max-von-Laue-Strasse 9, D-60438 Frankfurt am Main, Germany.
Curated by ChEMBL
Institute of Pharmaceutical Chemistry, Goethe-University Frankfurt , Max-von-Laue-Strasse 9, D-60438 Frankfurt am Main, Germany.
Curated by ChEMBL
Affinity DataKd: 1.22E+6nMAssay Description:Binding affinity to FXR (unknown origin)More data for this Ligand-Target Pair