Compile Data Set for Download or QSAR
Found 16 of ic50 data for polymerid = 2931
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
RIKEN

Curated by ChEMBL
LigandPNGBDBM50437341(WITHANOLIDE E)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8T7DPubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
RIKEN

Curated by ChEMBL
LigandPNGBDBM50437352(CHEMBL2408033)copy SMILEScopy InChI
Affinity DataIC50: 2.62E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8T7DPubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
RIKEN

Curated by ChEMBL
LigandPNGBDBM50378033(PHYSALIN F)copy SMILEScopy InChI
Affinity DataIC50: 2.71E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8T7DPubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
RIKEN

Curated by ChEMBL
LigandPNGBDBM50437349(25-HYDROXY PHYSALIN F)copy SMILEScopy InChI
Affinity DataIC50: 3.01E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8T7DPubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
RIKEN

Curated by ChEMBL
LigandPNGBDBM50378034(CHEMBL504404 | NSC-287088 | PHYSALIN B)copy SMILEScopy InChI
Affinity DataIC50: 3.75E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8T7DPubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
RIKEN

Curated by ChEMBL
LigandPNGBDBM50437346(CHEMBL2408037)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8T7DPubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
RIKEN

Curated by ChEMBL
LigandPNGBDBM50437347(PHYSALIN J)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8T7DPubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
RIKEN

Curated by ChEMBL
LigandPNGBDBM50437348(25-HYDROXY PHYSALIN J)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8T7DPubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
RIKEN

Curated by ChEMBL
LigandPNGBDBM50437350(CHEMBL2408034)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8T7DPubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
RIKEN

Curated by ChEMBL
LigandPNGBDBM50437351(PHYSALIN A)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8T7DPubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
RIKEN

Curated by ChEMBL
LigandPNGBDBM50437345(PHYSALIN O)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8T7DPubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
RIKEN

Curated by ChEMBL
LigandPNGBDBM50437344(WITHANOLIDE F)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8T7DPubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
RIKEN

Curated by ChEMBL
LigandPNGBDBM50437343(CHEMBL2333678)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8T7DPubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
RIKEN

Curated by ChEMBL
LigandPNGBDBM50437342(CHEMBL2333675)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8T7DPubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
RIKEN

Curated by ChEMBL
LigandPNGBDBM50437339(CHEMBL2408039)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8T7DPubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
RIKEN

Curated by ChEMBL
LigandPNGBDBM50437340(CHEMBL2408038)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8T7DPubMed