Compile Data Set for Download or QSAR
Found 13 of ic50 data for polymerid = 50001120
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
University College London

Curated by ChEMBL
LigandPNGBDBM50215069(1,2,3-tris-[3-(4-(N-ethyl)-quinoliniumylamino)-pro...)copy SMILEScopy InChI
Affinity DataIC50: 86nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416WSJPubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
University College London

Curated by ChEMBL
LigandPNGBDBM50215071(CHEMBL375272 | N-[3-(4-quinolinylamino)-propyl]-N-...)copy SMILEScopy InChI
Affinity DataIC50: 93nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416WSJPubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
University College London

Curated by ChEMBL
LigandPNGBDBM50215070(1,2,3-tri[3-(4-quinolinylamino)-propoxy]-benzene |...)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416WSJPubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
University College London

Curated by ChEMBL
LigandPNGBDBM50215076(CHEMBL229982 | N-[3-(4-quinolinylamino)-propyl]-N-...)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416WSJPubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
University College London

Curated by ChEMBL
LigandPNGBDBM50215075(CHEMBL229818 | N-[3-(4-quinolinylamino)-propyl]-3,...)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416WSJPubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
University College London

Curated by ChEMBL
LigandPNGBDBM50215072(CHEMBL389273 | N-(4-quinolinyl)-3,4-di-[3-(4-quino...)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416WSJPubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
University College London

Curated by ChEMBL
LigandPNGBDBM50215068(CHEMBL229341 | N-[3-(4-quinolinylamino)-proyl]-3,5...)copy SMILEScopy InChI
Affinity DataIC50: 360nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416WSJPubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
University College London

Curated by ChEMBL
LigandPNGBDBM50215073(CHEMBL229340 | N-[3-(4-quinolinyl)-aminopropyl]-N-...)copy SMILEScopy InChI
Affinity DataIC50: 490nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416WSJPubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
University College London

Curated by ChEMBL
LigandPNGBDBM50377980(CHEMBL558625)copy SMILEScopy InChI
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4QT0PubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
University College London

Curated by ChEMBL
LigandPNGBDBM50215074(CHEMBL425668 | N-(3-guanidinopropyl)-N-[4-(4'-amin...)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416WSJPubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
University College London

Curated by ChEMBL
LigandPNGBDBM50215079(4,4'bis(guanidinomethyl)-cis-stilbene | CHEMBL2291...)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416WSJPubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
University College London

Curated by ChEMBL
LigandPNGBDBM50215078(CHEMBL373955 | N-(3-guanidinopropyl)-N(8-aminoocty...)copy SMILEScopy InChI
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416WSJPubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rattus norvegicus)
University College London

Curated by ChEMBL
LigandPNGBDBM50215077(CHEMBL390821 | N-(3-guanidinopropyl)-N-(8-aminooct...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2416WSJPubMed