Compile Data Set for Download or QSAR
Found 17 of ki data for polymerid = 50001456
TargetMyeloblastin(Homo sapiens (Human))
INSERM UMR1100,"Centre d'Etude des Pathologies Respiratoires" , Université de Tours , 37032 Tours , France.

Curated by ChEMBL
LigandPNGBDBM50263166(CHEMBL4071346)copy SMILEScopy InChI
Affinity DataKi:  5.40nMAssay Description:Inhibition of human PR3 using ABZ-VADnVADYQ-EDDnp as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B04ZTPubMed
TargetMyeloblastin(Homo sapiens (Human))
INSERM UMR1100,"Centre d'Etude des Pathologies Respiratoires" , Université de Tours , 37032 Tours , France.

Curated by ChEMBL
LigandPNGBDBM50502655(CHEMBL4560512)copy SMILEScopy InChI
Affinity DataKi:  6.10nMAssay Description:Inhibition of purified human proteinase 3 using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58QNGPubMed
TargetMyeloblastin(Homo sapiens (Human))
INSERM UMR1100,"Centre d'Etude des Pathologies Respiratoires" , Université de Tours , 37032 Tours , France.

Curated by ChEMBL
LigandPNGBDBM50502658(CHEMBL4557877)copy SMILEScopy InChI
Affinity DataKi:  7nMAssay Description:Inhibition of purified human proteinase 3 using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58QNGPubMed
TargetMyeloblastin(Homo sapiens (Human))
INSERM UMR1100,"Centre d'Etude des Pathologies Respiratoires" , Université de Tours , 37032 Tours , France.

Curated by ChEMBL
LigandPNGBDBM50502659(CHEMBL4528256)copy SMILEScopy InChI
Affinity DataKi:  9.80nMAssay Description:Inhibition of purified human proteinase 3 using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58QNGPubMed
TargetMyeloblastin(Homo sapiens (Human))
INSERM UMR1100,"Centre d'Etude des Pathologies Respiratoires" , Université de Tours , 37032 Tours , France.

Curated by ChEMBL
LigandPNGBDBM50502656(CHEMBL4455694)copy SMILEScopy InChI
Affinity DataKi:  17nMAssay Description:Inhibition of purified human proteinase 3 using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58QNGPubMed
TargetMyeloblastin(Homo sapiens (Human))
INSERM UMR1100,"Centre d'Etude des Pathologies Respiratoires" , Université de Tours , 37032 Tours , France.

Curated by ChEMBL
LigandPNGBDBM50263172(CHEMBL4085013)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Inhibition of human PR3 using ABZ-VADnVADYQ-EDDnp as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B04ZTPubMed
TargetMyeloblastin(Homo sapiens (Human))
INSERM UMR1100,"Centre d'Etude des Pathologies Respiratoires" , Université de Tours , 37032 Tours , France.

Curated by ChEMBL
LigandPNGBDBM50502657(CHEMBL4589744)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Inhibition of purified human proteinase 3 using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58QNGPubMed
TargetMyeloblastin(Homo sapiens (Human))
INSERM UMR1100,"Centre d'Etude des Pathologies Respiratoires" , Université de Tours , 37032 Tours , France.

Curated by ChEMBL
LigandPNGBDBM50502654(CHEMBL4470455)copy SMILEScopy InChI
Affinity DataKi:  51nMAssay Description:Inhibition of purified human proteinase 3 using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58QNGPubMed
TargetMyeloblastin(Homo sapiens (Human))
INSERM UMR1100,"Centre d'Etude des Pathologies Respiratoires" , Université de Tours , 37032 Tours , France.

Curated by ChEMBL
LigandPNGBDBM50502660(CHEMBL4469546)copy SMILEScopy InChI
Affinity DataKi:  245nMAssay Description:Inhibition of purified human proteinase 3 using MeOSuc-AAPV-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58QNGPubMed
TargetMyeloblastin(Homo sapiens (Human))
INSERM UMR1100,"Centre d'Etude des Pathologies Respiratoires" , Université de Tours , 37032 Tours , France.

Curated by ChEMBL
LigandPNGBDBM50031630(CHEMBL3359765)copy SMILEScopy InChI
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of human PR3 using keto-D-DY-FRET as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ349FPubMed
TargetMyeloblastin(Homo sapiens (Human))
INSERM UMR1100,"Centre d'Etude des Pathologies Respiratoires" , Université de Tours , 37032 Tours , France.

Curated by ChEMBL
LigandPNGBDBM50263165(CHEMBL4102959)copy SMILEScopy InChI
Affinity DataKi:  3.60E+3nMAssay Description:Inhibition of human PR3 using ABZ-VADnVADYQ-EDDnp as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B04ZTPubMed
TargetMyeloblastin(Homo sapiens (Human))
INSERM UMR1100,"Centre d'Etude des Pathologies Respiratoires" , Université de Tours , 37032 Tours , France.

Curated by ChEMBL
LigandPNGBDBM50266984(CHEMBL4092637)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human PR3 using Suc(OMe)-AAPV-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB55DFPubMed
TargetMyeloblastin(Homo sapiens (Human))
INSERM UMR1100,"Centre d'Etude des Pathologies Respiratoires" , Université de Tours , 37032 Tours , France.

Curated by ChEMBL
LigandPNGBDBM50266979(CHEMBL4061897)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human PR3 using Suc(OMe)-AAPV-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB55DFPubMed
TargetMyeloblastin(Homo sapiens (Human))
INSERM UMR1100,"Centre d'Etude des Pathologies Respiratoires" , Université de Tours , 37032 Tours , France.

Curated by ChEMBL
LigandPNGBDBM50266989(CHEMBL4081142)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human PR3 using Suc(OMe)-AAPV-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB55DFPubMed
TargetMyeloblastin(Homo sapiens (Human))
INSERM UMR1100,"Centre d'Etude des Pathologies Respiratoires" , Université de Tours , 37032 Tours , France.

Curated by ChEMBL
LigandPNGBDBM247411(US10336754, Example 353 | US11053247, Example 353 ...)copy SMILEScopy InChI
Affinity DataKi: >1.20E+4nMAssay Description:Binding affinity to human neutrophil proteinase 3 assessed as inhibition constant using Methoxysuccinyl-L-alanyl-L-alanyl-L-prolylL-valine p-Nitroani...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20005Z7PubMed
TargetMyeloblastin(Homo sapiens (Human))
INSERM UMR1100,"Centre d'Etude des Pathologies Respiratoires" , Université de Tours , 37032 Tours , France.

Curated by ChEMBL
LigandPNGBDBM50544646(CHEMBL4635621)copy SMILEScopy InChI
Affinity DataKi:  2.65E+4nMAssay Description:Inhibition of human proteinase 3 using flurogenic substrate as elastase substrate V by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P357NPubMed
TargetMyeloblastin(Homo sapiens (Human))
INSERM UMR1100,"Centre d'Etude des Pathologies Respiratoires" , Université de Tours , 37032 Tours , France.

Curated by ChEMBL
LigandPNGBDBM50544648(CHEMBL4636971)copy SMILEScopy InChI
Affinity DataKi:  8.38E+4nMAssay Description:Inhibition of human proteinase 3 using flurogenic substrate as elastase substrate V by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P357NPubMed