Compile Data Set for Download or QSAR
Found 17 of ic50 data for polymerid = 50002441
TargetEndothelin-1 receptor(Mus musculus)
University Hospital M£nster

Curated by ChEMBL
LigandPNGBDBM50034267(3-(benzo[d][1,3]dioxol-5-yl)-5-hydroxy-5-(4-methox...)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Displacement of [125I]ET1 from endothelin A receptor in DBA mouse microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7NVFPubMed
TargetEndothelin-1 receptor(Mus musculus)
University Hospital M£nster

Curated by ChEMBL
LigandPNGBDBM50281579((S)-3-{2-[((R)-2-Acetylamino-3-phenyl-propionyl)-b...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27081C5
TargetEndothelin-1 receptor(Mus musculus)
University Hospital M£nster

Curated by ChEMBL
LigandPNGBDBM50281576((S)-3-{(S)-2-[(R)-2-Acetylamino-3-(1H-indol-3-yl)-...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27081C5
TargetEndothelin-1 receptor(Mus musculus)
University Hospital M£nster

Curated by ChEMBL
LigandPNGBDBM50281577((S)-3-{(S)-2-[(R)-2-Acetylamino-3-(4-hydroxy-pheny...)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27081C5
TargetEndothelin-1 receptor(Mus musculus)
University Hospital M£nster

Curated by ChEMBL
LigandPNGBDBM50281586((R)-3-{[(R)-1-((R)-2-Acetylamino-3-phenyl-propiony...)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27081C5
TargetEndothelin-1 receptor(Mus musculus)
University Hospital M£nster

Curated by ChEMBL
LigandPNGBDBM50281580((S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionyl...)copy SMILEScopy InChI
Affinity DataIC50: 57nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27081C5
TargetEndothelin-1 receptor(Mus musculus)
University Hospital M£nster

Curated by ChEMBL
LigandPNGBDBM50281581((S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionyl...)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27081C5
TargetEndothelin-1 receptor(Mus musculus)
University Hospital M£nster

Curated by ChEMBL
LigandPNGBDBM50281582((S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionyl...)copy SMILEScopy InChI
Affinity DataIC50: 75nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27081C5
TargetEndothelin-1 receptor(Mus musculus)
University Hospital M£nster

Curated by ChEMBL
LigandPNGBDBM50281575((S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionyl...)copy SMILEScopy InChI
Affinity DataIC50: 77nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27081C5
TargetEndothelin-1 receptor(Mus musculus)
University Hospital M£nster

Curated by ChEMBL
LigandPNGBDBM50281585((S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionyl...)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27081C5
TargetEndothelin-1 receptor(Mus musculus)
University Hospital M£nster

Curated by ChEMBL
LigandPNGBDBM50281587((S)-3-[(R)-2-((R)-2-Acetylamino-3-phenyl-propionyl...)copy SMILEScopy InChI
Affinity DataIC50: 98nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27081C5
TargetEndothelin-1 receptor(Mus musculus)
University Hospital M£nster

Curated by ChEMBL
LigandPNGBDBM50281583((S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionyl...)copy SMILEScopy InChI
Affinity DataIC50: 114nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27081C5
TargetEndothelin-1 receptor(Mus musculus)
University Hospital M£nster

Curated by ChEMBL
LigandPNGBDBM50281584((S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionyl...)copy SMILEScopy InChI
Affinity DataIC50: 230nMAssay Description:The compound was tested for the binding affinity against eEndothelin A receptor in murine 3T3 cells using [125I]-ET-1 as a radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27081C5
TargetEndothelin-1 receptor(Mus musculus)
University Hospital M£nster

Curated by ChEMBL
LigandPNGBDBM50281910((S)-3-[(S)-5-((S)-2-Acetylamino-3-phenyl-propionyl...)copy SMILEScopy InChI
Affinity DataIC50: 230nMAssay Description:Binding affinity of the compound for Endothelin A receptor was determined in murine 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC82S8
TargetEndothelin-1 receptor(Mus musculus)
University Hospital M£nster

Curated by ChEMBL
LigandPNGBDBM50281911((R)-3-[(R)-5-((S)-2-Acetylamino-3-phenyl-propionyl...)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Binding affinity of the compound for Endothelin A receptor was determined in murine 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC82S8
TargetEndothelin-1 receptor(Mus musculus)
University Hospital M£nster

Curated by ChEMBL
LigandPNGBDBM50281578((S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionyl...)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27081C5
TargetEndothelin-1 receptor(Mus musculus)
University Hospital M£nster

Curated by ChEMBL
LigandPNGBDBM50281912((S)-3-[(R)-5-((S)-2-Acetylamino-3-phenyl-propionyl...)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Binding affinity of the compound for Endothelin A receptor was determined in murine 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC82S8