TargetCyclin-dependent kinase 3/G1/S-specific cyclin-E1(Homo sapiens (Human))
H. Lee Moffitt Cancer Center and Research Institute
Curated by ChEMBL
H. Lee Moffitt Cancer Center and Research Institute
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Inhibition of CDK3/Cyclin E (unknown origin)-mediated phosphorylation of peptide substrate incubated for 15 mins prior to substrate addition measured...More data for this Ligand-Target Pair