Compile Data Set for Download or QSAR
Found 117 of ic50 data for polymerid = 50006164
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50581255(CHEMBL4531645)copy SMILES
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]-Tyr-Bpa-Ala-hexarelin from rat CD36 receptor in heart tissue membrane incubated for 60 mins by competitive receptor binding as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21RRPubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50581250(CHEMBL4455562)copy SMILES
Affinity DataIC50: 240nMAssay Description:Displacement of [125I]-Tyr-Bpa-Ala-hexarelin from rat CD36 receptor in heart tissue membrane incubated for 60 mins by competitive receptor binding as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21RRPubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50581260(CHEMBL4528721)copy SMILES
Affinity DataIC50: 670nMAssay Description:Displacement of [125I]-Tyr-Bpa-Ala-hexarelin from rat CD36 receptor in heart tissue membrane incubated for 60 mins by competitive receptor binding as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21RRPubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50581254(CHEMBL4471086)copy SMILES
Affinity DataIC50: 890nMAssay Description:Displacement of [125I]-Tyr-Bpa-Ala-hexarelin from rat CD36 receptor in heart tissue membrane incubated for 60 mins by competitive receptor binding as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21RRPubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50395009(CHEMBL2163470)copy SMILEScopy InChI
Affinity DataIC50: 1.11E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6D00PubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50395001(CHEMBL2163478 | US9708370, DBG-253-1)copy SMILEScopy InChI
Affinity DataIC50: 1.34E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6D00PubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50395001(CHEMBL2163478 | US9708370, DBG-253-1)copy SMILEScopy InChI
Affinity DataIC50: 1.34E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP76ZKUS Patent
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50370294(Examorelin | HEXARELIN | US9708370, Hexareline)copy SMILEScopy InChI
Affinity DataIC50: 1.56E+3nMAssay Description:Inhibition of photoactivatable [125I]-Tyr-Bpa-Ala-hexarelin binding to CD36 in Sprague-Dawley rat heart membranes after 60 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0WWVPubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50242203(CHEMBL4078128)copy SMILEScopy InChI
Affinity DataIC50: 1.65E+3nMAssay Description:Inhibition of photoactivatable [125I]-Tyr-Bpa-Ala-hexarelin binding to CD36 in Sprague-Dawley rat heart membranes after 60 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0WWVPubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50395007(CHEMBL2163472)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6D00PubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM263222(US9708370, DBG-175p)copy SMILES
Affinity DataIC50: 1.80E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP76ZKUS Patent
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50049479((S)-6-Amino-2-{(R)-2-[(S)-2-{(S)-2-[(R)-2-[(S)-2-a...)copy SMILEScopy InChI
Affinity DataIC50: 1.82E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6D00PubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50581259(CHEMBL5080816)copy SMILES
Affinity DataIC50: 1.86E+3nMAssay Description:Displacement of [125I]-Tyr-Bpa-Ala-hexarelin from rat CD36 receptor in heart tissue membrane incubated for 60 mins by competitive receptor binding as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21RRPubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50394994(CHEMBL2163484 | US9708370, DBG-178p)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of photoactivatable [125I]-Tyr-Bpa-Ala-hexarelin binding to CD36 in Sprague-Dawley rat heart membranes after 60 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0WWVPubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50370294(Examorelin | HEXARELIN | US9708370, Hexareline)copy SMILEScopy InChI
Affinity DataIC50: 2.08E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6D00PubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50581261(CHEMBL5092625)copy SMILES
Affinity DataIC50: 2.26E+3nMAssay Description:Displacement of [125I]-Tyr-Bpa-Ala-hexarelin from rat CD36 receptor in heart tissue membrane incubated for 60 mins by competitive receptor binding as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21RRPubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50395002(CHEMBL2163477 | US9708370, DBG-201-A)copy SMILEScopy InChI
Affinity DataIC50: 2.89E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6D00PubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50395002(CHEMBL2163477 | US9708370, DBG-201-A)copy SMILEScopy InChI
Affinity DataIC50: 2.89E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP76ZKUS Patent
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM263256(US9708370, 67 ZS555-F40 | US9708370, ZS555-F40)copy SMILES
Affinity DataIC50: 2.95E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP76ZKUS Patent
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50370294(Examorelin | HEXARELIN | US9708370, Hexareline)copy SMILEScopy InChI
Affinity DataIC50: 2.97E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP76ZKUS Patent
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50581258(CHEMBL5094226)copy SMILES
Affinity DataIC50: 3.06E+3nMAssay Description:Displacement of [125I]-Tyr-Bpa-Ala-hexarelin from rat CD36 receptor in heart tissue membrane incubated for 60 mins by competitive receptor binding as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21RRPubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50370294(Examorelin | HEXARELIN | US9708370, Hexareline)copy SMILEScopy InChI
Affinity DataIC50: 3.33E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP76ZKUS Patent
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50242204(CHEMBL4086017)copy SMILEScopy InChI
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of HIV-1 protease in 10% fetal calf serum(FCS)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0WWVPubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50395019(CHEMBL2163449 | US9708370, CP-2B(v))copy SMILEScopy InChI
Affinity DataIC50: 3.68E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP76ZKUS Patent
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50581256(CHEMBL5087491)copy SMILES
Affinity DataIC50: 4.75E+3nMAssay Description:Displacement of [125I]-Tyr-Bpa-Ala-hexarelin from rat CD36 receptor in heart tissue membrane incubated for 60 mins by competitive receptor binding as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21RRPubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50395016(CHEMBL2163452 | US9708370, CP-2B(ii))copy SMILEScopy InChI
Affinity DataIC50: 4.94E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP76ZKUS Patent
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50242206(CHEMBL4080592)copy SMILEScopy InChI
Affinity DataIC50: 4.94E+3nMAssay Description:Inhibition of photoactivatable [125I]-Tyr-Bpa-Ala-hexarelin binding to CD36 in Sprague-Dawley rat heart membranes after 60 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0WWVPubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50394993(CHEMBL2163485 | US9708370, CP-1A(iv))copy SMILEScopy InChI
Affinity DataIC50: 5.02E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP76ZKUS Patent
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50242210(CHEMBL4104823)copy SMILEScopy InChI
Affinity DataIC50: 5.51E+3nMAssay Description:Inhibition of photoactivatable [125I]-Tyr-Bpa-Ala-hexarelin binding to CD36 in Sprague-Dawley rat heart membranes after 60 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0WWVPubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50242216(CHEMBL4088461)copy SMILEScopy InChI
Affinity DataIC50: 5.58E+3nMAssay Description:Inhibition of HIV-1 protease in 10% fetal calf serum(FCS)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0WWVPubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50395024(CHEMBL2163444 | US9708370, CP-2A(v))copy SMILEScopy InChI
Affinity DataIC50: 6.06E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6D00PubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50242211(CHEMBL4067202)copy SMILEScopy InChI
Affinity DataIC50: 6.06E+3nMAssay Description:Inhibition of photoactivatable [125I]-Tyr-Bpa-Ala-hexarelin binding to CD36 in Sprague-Dawley rat heart membranes after 60 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0WWVPubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50395019(CHEMBL2163449 | US9708370, CP-2B(v))copy SMILEScopy InChI
Affinity DataIC50: 6.66E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6D00PubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50242212(CHEMBL4085058)copy SMILEScopy InChI
Affinity DataIC50: 7.51E+3nMAssay Description:Inhibitory concentration against HIV-2 protease in the absence of DMSOMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0WWVPubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50395014(CHEMBL2163454 | US9708370, 60 CP-3(iv))copy SMILEScopy InChI
Affinity DataIC50: 7.58E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6D00PubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50395015(CHEMBL2163453 | US9708370, CP-2B(i))copy SMILEScopy InChI
Affinity DataIC50: 7.59E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6D00PubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50394983(CHEMBL2163466)copy SMILEScopy InChI
Affinity DataIC50: 7.97E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6D00PubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50242213(CHEMBL4063430)copy SMILEScopy InChI
Affinity DataIC50: 8.36E+3nMAssay Description:Inhibition of HIV-1 protease in 10% fetal calf serum(FCS)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0WWVPubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50395024(CHEMBL2163444 | US9708370, CP-2A(v))copy SMILEScopy InChI
Affinity DataIC50: 8.76E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP76ZKUS Patent
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50394982(CHEMBL2163467)copy SMILEScopy InChI
Affinity DataIC50: 9.01E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6D00PubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50395015(CHEMBL2163453 | US9708370, CP-2B(i))copy SMILEScopy InChI
Affinity DataIC50: 9.02E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP76ZKUS Patent
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50581262(CHEMBL5086116)copy SMILES
Affinity DataIC50: 9.05E+3nMAssay Description:Displacement of [125I]-Tyr-Bpa-Ala-hexarelin from rat CD36 receptor in heart tissue membrane incubated for 60 mins by competitive receptor binding as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21RRPubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM263256(US9708370, 67 ZS555-F40 | US9708370, ZS555-F40)copy SMILES
Affinity DataIC50: 9.19E+3nMAssay Description:Inhibition of photoactivatable [125I]-Tyr-Bpa-Ala-hexarelin binding to CD36 in Sprague-Dawley rat heart membranes after 60 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0WWVPubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50395016(CHEMBL2163452 | US9708370, CP-2B(ii))copy SMILEScopy InChI
Affinity DataIC50: 9.48E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6D00PubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50395003(CHEMBL2163476 | US9708370, DBG-188p)copy SMILEScopy InChI
Affinity DataIC50: 9.61E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6D00PubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50395003(CHEMBL2163476 | US9708370, DBG-188p)copy SMILEScopy InChI
Affinity DataIC50: 9.61E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP76ZKUS Patent
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50395017(CHEMBL2163451 | US9708370, CP-2B(iii))copy SMILEScopy InChI
Affinity DataIC50: 9.66E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP76ZKUS Patent
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50394989(CHEMBL2163460 | US9708370, 62 CP-AP-4)copy SMILEScopy InChI
Affinity DataIC50: 9.81E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6D00PubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50394991(CHEMBL2163438 | US9708370, 40 CP-1A(ii))copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6D00PubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)TBA
LigandPNGBDBM50394992(CHEMBL2163437)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6D00PubMed
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