Compile Data Set for Download or QSAR
Found 125 of ec50 data for polymerid = 50006785
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50085928(CHEMBL3425593)copy SMILEScopy InChI
Affinity DataEC50:  0.0830nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as intracellular calcium flux at by Fluo-4 AM dye based fluorometric imaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CVPPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049421(CHEMBL3315349)copy SMILEScopy InChI
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as intracellular calcium flux at by Fluo-4 AM dye based fluorometric imaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CVPPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50239755(CHEMBL4069151)copy SMILEScopy InChI
Affinity DataEC50:  0.170nMAssay Description:Antisecretory activity evaluated by the inhibition of 14C -AP uptake in isolated rabbit parietal cells stimulated by exogenous histamineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46V4JPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50239756(CHEMBL4105671)copy SMILEScopy InChI
Affinity DataEC50:  0.25nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux after 18 hrs by Fluo-4 AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46V4JPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50238694(CHEMBL4098010)copy SMILEScopy InChI
Affinity DataEC50:  0.310nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux measured for 180 secs by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37ZKKPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50238690(CHEMBL4068681)copy SMILEScopy InChI
Affinity DataEC50:  0.320nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux measured for 180 secs by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37ZKKPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50238691(CHEMBL4088263)copy SMILEScopy InChI
Affinity DataEC50:  0.410nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux measured for 180 secs by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37ZKKPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049421(CHEMBL3315349)copy SMILEScopy InChI
Affinity DataEC50:  0.430nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FQ9Z71PubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049425(CHEMBL3356083)copy SMILEScopy InChI
Affinity DataEC50:  0.450nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as increase in intracellular calcium influx after 180 secs by Fluo 4-AM dye based FLI...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HMNPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50291730(CHEMBL4169726)copy SMILEScopy InChI
Affinity DataEC50:  0.510nMAssay Description:Agonist activity at human NMUR1 expressed in HEK293 cells assessed as IP3 accumulation after 60 mins in presence of myo-[2-3H(N)]inositol by scintill...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB55HSPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50291730(CHEMBL4169726)copy SMILEScopy InChI
Affinity DataEC50:  0.510nMAssay Description:Agonist activity at human NMUR1 expressed in HEK293 cells assessed as induction of IP3 levels using myo-[2-3H(N)]-inositol after 60 mins by SPA-based...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B91JPPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049425(CHEMBL3356083)copy SMILEScopy InChI
Affinity DataEC50:  0.540nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux measured for 180 secs by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37ZKKPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50500779(CHEMBL3758577)copy SMILEScopy InChI
Affinity DataEC50:  0.562nMAssay Description:Agonist activity at recombinant human NMU1 expressed in HEK293 cells assessed as change in intracellular calcium flux by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26H4MFFPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50500783(CHEMBL3759452)copy SMILEScopy InChI
Affinity DataEC50:  0.575nMAssay Description:Agonist activity at recombinant human NMU1 expressed in HEK293 cells assessed as change in intracellular calcium flux by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26H4MFFPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50238707(CHEMBL4059530)copy SMILEScopy InChI
Affinity DataEC50:  0.730nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux measured for 180 secs by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37ZKKPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50238689(CHEMBL4073946)copy SMILEScopy InChI
Affinity DataEC50:  0.770nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux measured for 180 secs by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37ZKKPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50238704(CHEMBL4095998)copy SMILEScopy InChI
Affinity DataEC50:  0.960nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux measured for 180 secs by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37ZKKPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50238695(CHEMBL4079986)copy SMILEScopy InChI
Affinity DataEC50:  1nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux measured for 180 secs by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37ZKKPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049421(CHEMBL3315349)copy SMILEScopy InChI
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at recombinant human NMU1 expressed in HEK293 cells assessed as change in intracellular calcium flux by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26H4MFFPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50238693(CHEMBL4063830)copy SMILEScopy InChI
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux measured for 180 secs by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37ZKKPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50291716(CHEMBL4161902)copy SMILEScopy InChI
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at human NMUR1 expressed in HEK293 cells assessed as induction of IP3 levels using myo-[2-3H(N)]-inositol after 60 mins by SPA-based...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B91JPPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049424(CHEMBL3315348)copy SMILEScopy InChI
Affinity DataEC50:  1.70nMAssay Description:Partial agonist activity at human NMUR1 expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC077ZPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50500784(CHEMBL4299242)copy SMILEScopy InChI
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at recombinant human NMU1 expressed in HEK293 cells assessed as change in intracellular calcium flux by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26H4MFFPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50238696(CHEMBL4087867)copy SMILEScopy InChI
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux measured for 180 secs by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37ZKKPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049424(CHEMBL3315348)copy SMILEScopy InChI
Affinity DataEC50:  2.20nMAssay Description:Partial agonist activity at human NMUR1 expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FQ9Z71PubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50238701(CHEMBL4061507)copy SMILEScopy InChI
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux measured for 180 secs by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37ZKKPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50238706(CHEMBL4099780)copy SMILEScopy InChI
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux measured for 180 secs by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37ZKKPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50238700(CHEMBL4089636)copy SMILEScopy InChI
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux measured for 180 secs by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37ZKKPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50338535(CHEMBL4162728)copy SMILEScopy InChI
Affinity DataEC50:  2.90nMAssay Description:Agonist activity at human NMUR1 expressed in HEK293 cells assessed as IP3 accumulation after 60 mins in presence of myo-[2-3H(N)]inositol by scintill...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB55HSPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50560260(CHEMBL4798983)copy SMILES
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC077ZPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50336621(CHEMBL4170275)copy SMILEScopy InChI
Affinity DataEC50:  3.70nMAssay Description:Agonist activity at human NMUR1 expressed in HEK293 cells assessed as IP3 accumulation after 60 mins in presence of myo-[2-3H(N)]inositol by scintill...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB55HSPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50291714(CHEMBL4177021)copy SMILEScopy InChI
Affinity DataEC50:  4nMAssay Description:Agonist activity at human NMUR1 expressed in HEK293 cells assessed as induction of IP3 levels using myo-[2-3H(N)]-inositol after 60 mins by SPA-based...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B91JPPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50291699(CHEMBL4175546)copy SMILEScopy InChI
Affinity DataEC50:  4.20nMAssay Description:Agonist activity at human NMUR1 expressed in HEK293 cells assessed as induction of IP3 levels using myo-[2-3H(N)]-inositol after 60 mins by SPA-based...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B91JPPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50291701(CHEMBL4165337)copy SMILEScopy InChI
Affinity DataEC50:  4.30nMAssay Description:Agonist activity at human NMUR1 expressed in HEK293 cells assessed as induction of IP3 levels using myo-[2-3H(N)]-inositol after 60 mins by SPA-based...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B91JPPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50291718(CHEMBL4174679)copy SMILEScopy InChI
Affinity DataEC50:  5.10nMAssay Description:Agonist activity at human NMUR1 expressed in HEK293 cells assessed as induction of IP3 levels using myo-[2-3H(N)]-inositol after 60 mins by SPA-based...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B91JPPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50291719(CHEMBL4165538)copy SMILEScopy InChI
Affinity DataEC50:  5.5nMAssay Description:Agonist activity at human NMUR1 expressed in HEK293 cells assessed as induction of IP3 levels using myo-[2-3H(N)]-inositol after 60 mins by SPA-based...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B91JPPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50262111(CHEMBL4081819)copy SMILEScopy InChI
Affinity DataEC50:  6.30nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as increase in intracellular calcium influx after 180 secs by Fluo 4-AM dye based FLI...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HMNPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50291696(CHEMBL4164922)copy SMILEScopy InChI
Affinity DataEC50:  7.70nMAssay Description:Agonist activity at human NMUR1 expressed in HEK293 cells assessed as induction of IP3 levels using myo-[2-3H(N)]-inositol after 60 mins by SPA-based...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B91JPPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50238710(CHEMBL4091611)copy SMILEScopy InChI
Affinity DataEC50:  7.80nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux measured for 180 secs by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37ZKKPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50291727(CHEMBL4175315)copy SMILEScopy InChI
Affinity DataEC50:  8.10nMAssay Description:Agonist activity at human NMUR1 expressed in HEK293 cells assessed as induction of IP3 levels using myo-[2-3H(N)]-inositol after 60 mins by SPA-based...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B91JPPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50238711(CHEMBL4097355)copy SMILEScopy InChI
Affinity DataEC50:  8.10nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux measured for 180 secs by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37ZKKPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049423(CHEMBL3315278)copy SMILEScopy InChI
Affinity DataEC50:  9nMAssay Description:Partial agonist activity at human NMUR1 expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FQ9Z71PubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50238703(CHEMBL4081760)copy SMILEScopy InChI
Affinity DataEC50:  9.20nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux measured for 180 secs by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37ZKKPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50262099(CHEMBL4074121)copy SMILEScopy InChI
Affinity DataEC50:  9.5nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as increase in intracellular calcium influx after 180 secs by Fluo 4-AM dye based FLI...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0HMNPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50238699(CHEMBL4063341)copy SMILEScopy InChI
Affinity DataEC50:  9.5nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux measured for 180 secs by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37ZKKPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50291715(CHEMBL4172552)copy SMILEScopy InChI
Affinity DataEC50:  10nMAssay Description:Agonist activity at human NMUR1 expressed in HEK293 cells assessed as induction of IP3 levels using myo-[2-3H(N)]-inositol after 60 mins by SPA-based...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B91JPPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50336637(CHEMBL4159554)copy SMILEScopy InChI
Affinity DataEC50:  11nMAssay Description:Agonist activity at human NMUR1 expressed in HEK293 cells assessed as IP3 accumulation after 60 mins in presence of myo-[2-3H(N)]inositol by scintill...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB55HSPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50291731(CHEMBL4168753)copy SMILEScopy InChI
Affinity DataEC50:  12nMAssay Description:Agonist activity at human NMUR1 expressed in HEK293 cells assessed as induction of IP3 levels using myo-[2-3H(N)]-inositol after 60 mins by SPA-based...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B91JPPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50500776(CHEMBL3759206)copy SMILEScopy InChI
Affinity DataEC50:  12nMAssay Description:Agonist activity at recombinant human NMU1 expressed in HEK293 cells assessed as change in intracellular calcium flux by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26H4MFFPubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50238697(CHEMBL4090300)copy SMILEScopy InChI
Affinity DataEC50:  17nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux measured for 180 secs by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37ZKKPubMed
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