Compile Data Set for Download or QSAR
Found 150 of ic50 data for polymerid = 50006865,8828
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50005782(ATI-13387X | ONALESPIB)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ72FHPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50180302(8-(6-iodo-benzo[1,3]dioxol-5-ylsulfanyl)-9-(3-isop...)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50087812(CHEMBL3426787)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of GRP94 (unknown origin) expressed in HEK293 cells assessed as reduction of Toll-like receptor trafficking to cell membrane treated for 2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2CSDPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50439621(GANETESPIB | STA-9090)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1W9TPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50540240(CHEMBL4647894)copy SMILEScopy InChI
Affinity DataIC50: 49nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1W9TPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50555415(CHEMBL4744238)copy SMILES
Affinity DataIC50: 50nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ72FHPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50540237(CHEMBL4647171)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1W9TPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50540239(CHEMBL4635982)copy SMILEScopy InChI
Affinity DataIC50: 78nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1W9TPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50540232(CHEMBL4641526)copy SMILEScopy InChI
Affinity DataIC50: 78nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1W9TPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM20926(5-[2,4-dihydroxy-5-(propan-2-yl)phenyl]-N-ethyl-4-...)copy SMILEScopy InChI
Affinity DataIC50: 85nMAssay Description:Inhibition of Grp94More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM889JPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50540236(CHEMBL4639163)copy SMILEScopy InChI
Affinity DataIC50: 89nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1W9TPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50540249(CHEMBL4635778)copy SMILEScopy InChI
Affinity DataIC50: 96nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1W9TPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50540248(CHEMBL4648197)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1W9TPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50087810(CHEMBL3426784 | US10428068, Compound 52 | US108440...)copy SMILEScopy InChI
Affinity DataIC50: 101nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50165316(8-(2,4-Dichloro-phenylsulfanyl)-9-pent-4-ynyl-9H-p...)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50180302(8-(6-iodo-benzo[1,3]dioxol-5-ylsulfanyl)-9-(3-isop...)copy SMILEScopy InChI
Affinity DataIC50: 132nMAssay Description:Inhibition of PU-H71-FITC3 binding to recombinant N-terminal Grp94 (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G164M9PubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50165315(9-Pent-4-ynyl-8-(2,4,5-trichloro-phenylsulfanyl)-9...)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50540242(CHEMBL4648091)copy SMILEScopy InChI
Affinity DataIC50: 175nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1W9TPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50540238(CHEMBL4638275)copy SMILEScopy InChI
Affinity DataIC50: 190nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1W9TPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50540251(CHEMBL4641450)copy SMILEScopy InChI
Affinity DataIC50: 192nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1W9TPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50571896(CHEMBL4869481)copy SMILES
Affinity DataIC50: 194nMAssay Description:Inhibition of PU-H71-FITC3 binding to recombinant N-terminal Grp94 (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G164M9PubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50555456(CHEMBL4779990)copy SMILES
Affinity DataIC50: 195nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ72FHPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50555451(CHEMBL4782374)copy SMILES
Affinity DataIC50: 196nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ72FHPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50540241(CHEMBL4636983)copy SMILEScopy InChI
Affinity DataIC50: 197nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1W9TPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50555440(CHEMBL4797602)copy SMILES
Affinity DataIC50: 198nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ72FHPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50540250(CHEMBL4649532)copy SMILEScopy InChI
Affinity DataIC50: 209nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1W9TPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50555455(CHEMBL4753741)copy SMILES
Affinity DataIC50: 216nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ72FHPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50555442(CHEMBL4777147)copy SMILES
Affinity DataIC50: 217nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ72FHPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50087721(CHEMBL3426781)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50555447(CHEMBL4753836)copy SMILES
Affinity DataIC50: 232nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ72FHPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50087447(CHEMBL3426734)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50555416(CHEMBL4781723)copy SMILES
Affinity DataIC50: 245nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ72FHPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50165268(8-(3,5-Dichloro-phenylsulfanyl)-9-pent-4-ynyl-9H-p...)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50087811(CHEMBL3426785)copy SMILEScopy InChI
Affinity DataIC50: 265nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50087454(CHEMBL3426741)copy SMILEScopy InChI
Affinity DataIC50: 287nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50555441(CHEMBL4744192)copy SMILES
Affinity DataIC50: 290nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ72FHPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50087448(CHEMBL3426735)copy SMILEScopy InChI
Affinity DataIC50: 290nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50180302(8-(6-iodo-benzo[1,3]dioxol-5-ylsulfanyl)-9-(3-isop...)copy SMILEScopy InChI
Affinity DataIC50: 301nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1W9TPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50571903(CHEMBL4863672)copy SMILES
Affinity DataIC50: 318nMAssay Description:Inhibition of PU-H71-FITC3 binding to recombinant N-terminal Grp94 (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G164M9PubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50087575(CHEMBL3426763)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50165295(8-(2-Chloro-phenylsulfanyl)-9-pent-4-ynyl-9H-purin...)copy SMILEScopy InChI
Affinity DataIC50: 350nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50087524(CHEMBL3426756)copy SMILEScopy InChI
Affinity DataIC50: 390nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50087445(CHEMBL3426733)copy SMILEScopy InChI
Affinity DataIC50: 390nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50087720(CHEMBL3426780)copy SMILEScopy InChI
Affinity DataIC50: 410nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50087507(CHEMBL3426748)copy SMILEScopy InChI
Affinity DataIC50: 429nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50087452(CHEMBL3426739)copy SMILEScopy InChI
Affinity DataIC50: 430nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC12DDPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50240873(CHEMBL4068596)copy SMILEScopy InChI
Affinity DataIC50: 448nMAssay Description:Inhibition of PU-H71-FITC3 binding to recombinant N-terminal Grp94 (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G164M9PubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50571897(CHEMBL4866705)copy SMILES
Affinity DataIC50: 494nMAssay Description:Inhibition of PU-H71-FITC3 binding to recombinant N-terminal Grp94 (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G164M9PubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50555432(CHEMBL4757080)copy SMILES
Affinity DataIC50: 498nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ72FHPubMed
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM50555430(CHEMBL4778735)copy SMILES
Affinity DataIC50: 498nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ72FHPubMed
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