Compile Data Set for Download or QSAR
Found 6 of ic50 for UniProtKB: P26818
TargetBeta-adrenergic receptor kinase 2(Bos taurus)
Universit£ degli Studi di Messina

Curated by ChEMBL
LigandPNGBDBM50191311(CHEMBL3950887)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of recombinant bovine GRK3 expressed in Sf9 insect cells assessed as decrease in phosphorylation of urea-washed bovine rod outer segments ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2348NB9PubMed
TargetBeta-adrenergic receptor kinase 2(Bos taurus)
Universit£ degli Studi di Messina

Curated by ChEMBL
LigandPNGBDBM50191313(CHEMBL3931500)copy SMILEScopy InChI
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of recombinant bovine GRK3 expressed in Sf9 insect cells assessed as decrease in phosphorylation of urea-washed bovine rod outer segments ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2348NB9PubMed
TargetBeta-adrenergic receptor kinase 2(Bos taurus)
Universit£ degli Studi di Messina

Curated by ChEMBL
LigandPNGBDBM50191319(CHEMBL3942164)copy SMILEScopy InChI
Affinity DataIC50: 1.16E+4nMAssay Description:Inhibition of recombinant bovine GRK3 expressed in Sf9 insect cells assessed as decrease in phosphorylation of urea-washed bovine rod outer segments ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2348NB9PubMed
TargetBeta-adrenergic receptor kinase 2(Bos taurus)
Universit£ degli Studi di Messina

Curated by ChEMBL
LigandPNGBDBM50191326(CHEMBL3953837)copy SMILEScopy InChI
Affinity DataIC50: 2.26E+4nMAssay Description:Inhibition of recombinant bovine GRK3 expressed in Sf9 insect cells assessed as decrease in phosphorylation of urea-washed bovine rod outer segments ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2348NB9PubMed
TargetBeta-adrenergic receptor kinase 2(Bos taurus)
Universit£ degli Studi di Messina

Curated by ChEMBL
LigandPNGBDBM50191312(CHEMBL3900757)copy SMILEScopy InChI
Affinity DataIC50: 3.04E+4nMAssay Description:Inhibition of recombinant bovine GRK3 expressed in Sf9 insect cells assessed as decrease in phosphorylation of urea-washed bovine rod outer segments ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2348NB9PubMed
TargetBeta-adrenergic receptor kinase 2(Bos taurus)
Universit£ degli Studi di Messina

Curated by ChEMBL
LigandPNGBDBM50191310(CHEMBL3971763)copy SMILEScopy InChI
Affinity DataIC50: 5.55E+4nMAssay Description:Inhibition of recombinant bovine GRK3 expressed in Sf9 insect cells assessed as decrease in phosphorylation of urea-washed bovine rod outer segments ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2348NB9PubMed