Compile Data Set for Download or QSAR
Found 12 of ki data for polymerid = 50007165
TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
GTx, Inc.; THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS

US Patent
LigandPNGBDBM312140(6,8-dihydroxy-2-(4-hydroxyphenyl)-4-(4-methoxyphen...)copy SMILEScopy InChI
Affinity DataKi:  0.480nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N25FRUS Patent
TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
GTx, Inc.; THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS

US Patent
LigandPNGBDBM312151((E)-6,8-dihydroxy-2-(4-hydroxyphenyl)-4-(prop-1-en...)copy SMILEScopy InChI
Affinity DataKi:  1.66nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N25FRUS Patent
TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
GTx, Inc.; THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS

US Patent
LigandPNGBDBM312096(4-bromo-6,8-dihydroxy-2-(4-hydroxyphenyl)isoquinol...)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N25FRUS Patent
TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
GTx, Inc.; THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS

US Patent
LigandPNGBDBM312133(US9604931, 12z)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N25FRUS Patent
TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
GTx, Inc.; THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS

US Patent
LigandPNGBDBM312149(6,8-dihydroxy-2-(4-hydroxyphenyl)-4-(4-methoxyphen...)copy SMILEScopy InChI
Affinity DataKi:  3.03nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N25FRUS Patent
TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
GTx, Inc.; THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS

US Patent
LigandPNGBDBM312139(2-(3-fluoro-4-hydroxyphenyl)-6,8-dihydroxy-4-vinyl...)copy SMILEScopy InChI
Affinity DataKi:  3.96nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N25FRUS Patent
TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
GTx, Inc.; THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS

US Patent
LigandPNGBDBM312134(4-bromo-6-methoxy-2-(4-methoxyphenyl)-1-oxo-1,2-di...)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N25FRUS Patent
TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
GTx, Inc.; THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS

US Patent
LigandPNGBDBM312135(6,8-dihydroxy-2-(4-hydroxyphenyl)-1-oxo-1,2-dihydr...)copy SMILEScopy InChI
Affinity DataKi:  7nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N25FRUS Patent
TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
GTx, Inc.; THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS

US Patent
LigandPNGBDBM312136(4-bromo-6-hydroxy-2-(4-hydroxyphenyl)-1-oxo-1,2-di...)copy SMILEScopy InChI
Affinity DataKi:  46nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N25FRUS Patent
TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
GTx, Inc.; THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS

US Patent
LigandPNGBDBM310198(4-bromo-6-hydroxy-2-(4-hydroxyphenyl)isoquinolin-1...)copy SMILEScopy InChI
Affinity DataKi:  49nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N25FRUS Patent
TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
GTx, Inc.; THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS

US Patent
LigandPNGBDBM312137(6-hydroxy-2-(4-hydroxyphenyl)-4-phenylisoquinolin-...)copy SMILEScopy InChI
Affinity DataKi:  130nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N25FRUS Patent
TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
GTx, Inc.; THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS

US Patent
LigandPNGBDBM312138(6-hydroxy-2-(4-hydroxyphenol)-4-(4-methoxyphenyl)i...)copy SMILEScopy InChI
Affinity DataKi:  252nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23N25FRUS Patent