Compile Data Set for Download or QSAR
Found 74 of ic50 data for polymerid = 9048
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092072(CHEMBL3582419 | US9296728, 14)copy SMILEScopy InChI
Affinity DataIC50: 7.60nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0M5RUS Patent
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092069(CHEMBL3582422 | US9296728, 20)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84MVPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092069(CHEMBL3582422 | US9296728, 20)copy SMILEScopy InChI
Affinity DataIC50: 8nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0M5RUS Patent
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092072(CHEMBL3582419 | US9296728, 14)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84MVPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092073(CHEMBL3582418 | US9296728, 13)copy SMILEScopy InChI
Affinity DataIC50: 9.5nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0M5RUS Patent
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092058(CHEMBL3582408)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84MVPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092071(CHEMBL3582420 | US9296728, 18)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84MVPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092068(CHEMBL3582423)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84MVPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092073(CHEMBL3582418 | US9296728, 13)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84MVPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50608638(CHEMBL4303684)copy SMILES
Affinity DataIC50: 13nMMore data for this Ligand-Target Pair
Ligand InfoPDB
In DepthDetails
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092071(CHEMBL3582420 | US9296728, 18)copy SMILEScopy InChI
Affinity DataIC50: 15nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0M5RUS Patent
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM214697(US9296728, 19)copy SMILEScopy InChI
Affinity DataIC50: 19nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0M5RUS Patent
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092070(CHEMBL3582421 | US9296728, 15)copy SMILEScopy InChI
Affinity DataIC50: 23nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0M5RUS Patent
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092067(CHEMBL3582424 | US9296728, 16)copy SMILEScopy InChI
Affinity DataIC50: 25nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0M5RUS Patent
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092065(CHEMBL3582426)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84MVPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092057(CHEMBL3582409 | US9296728, 4)copy SMILEScopy InChI
Affinity DataIC50: 26nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0M5RUS Patent
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092067(CHEMBL3582424 | US9296728, 16)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84MVPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092057(CHEMBL3582409 | US9296728, 4)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84MVPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092076(CHEMBL3582415)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84MVPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092070(CHEMBL3582421 | US9296728, 15)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84MVPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM214695(US9296728, 10)copy SMILEScopy InChI
Affinity DataIC50: 43nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0M5RUS Patent
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM214702(US9296728, 25)copy SMILEScopy InChI
Affinity DataIC50: 48nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0M5RUS Patent
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092066(CHEMBL3582425)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84MVPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM214698(US9296728, 21)copy SMILEScopy InChI
Affinity DataIC50: 59nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0M5RUS Patent
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092075(CHEMBL3582416 | US9296728, 11)copy SMILEScopy InChI
Affinity DataIC50: 64nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0M5RUS Patent
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50606661(CHEMBL5220706)copy SMILES
Affinity DataIC50: 66nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61QBTPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50608639(CHEMBL4793546)copy SMILES
Affinity DataIC50: 66nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092018(CHEMBL3582410 | US9296728, 9)copy SMILEScopy InChI
Affinity DataIC50: 66nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0M5RUS Patent
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092075(CHEMBL3582416 | US9296728, 11)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84MVPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092059(CHEMBL3582407)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84MVPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092078(CHEMBL3582413 | US9296728, 7)copy SMILEScopy InChI
Affinity DataIC50: 88nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0M5RUS Patent
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM214702(US9296728, 25)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of MCT1 in rat brain endothelial 4 cells assessed as L-[14C]-Lactate Uptake after 15 mins by scintillation spectrometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP04QPPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM214696(US9296728, 17)copy SMILEScopy InChI
Affinity DataIC50: 91nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0M5RUS Patent
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50608637(CHEMBL5280660)copy SMILES
Affinity DataIC50: 97nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092018(CHEMBL3582410 | US9296728, 9)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84MVPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM214705(US9296728, 29)copy SMILEScopy InChI
Affinity DataIC50: 110nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0M5RUS Patent
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092074(CHEMBL3582417 | US9296728, 12)copy SMILEScopy InChI
Affinity DataIC50: 110nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0M5RUS Patent
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092078(CHEMBL3582413 | US9296728, 7)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84MVPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092017(CHEMBL3582411 | US9296728, 5)copy SMILEScopy InChI
Affinity DataIC50: 120nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0M5RUS Patent
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092017(CHEMBL3582411 | US9296728, 5)copy SMILEScopy InChI
Affinity DataIC50: 140nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84MVPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50092074(CHEMBL3582417 | US9296728, 12)copy SMILEScopy InChI
Affinity DataIC50: 140nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84MVPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM4345((2E)-2-cyano-3-[4-(dimethylamino)phenyl]prop-2-eno...)copy SMILEScopy InChI
Affinity DataIC50: 140nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84MVPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM214701(US9296728, 24)copy SMILEScopy InChI
Affinity DataIC50: 150nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0M5RUS Patent
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM214700(US9296728, 23)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Inhibition of MCT1 in rat brain endothelial 4 cells assessed as L-[14C]-Lactate Uptake after 15 mins by scintillation spectrometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP04QPPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM214703(US9296728, 27)copy SMILEScopy InChI
Affinity DataIC50: 200nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0M5RUS Patent
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM214701(US9296728, 24)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Inhibition of MCT1 in rat brain endothelial 4 cells assessed as L-[14C]-Lactate Uptake after 15 mins by scintillation spectrometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP04QPPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM50442702(CHEMBL2442511 | US9296728, 26)copy SMILEScopy InChI
Affinity DataIC50: 220nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0M5RUS Patent
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM214700(US9296728, 23)copy SMILEScopy InChI
Affinity DataIC50: 250nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0M5RUS Patent
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM4350((2E)-2-cyano-3-(4-hydroxyphenyl)prop-2-enoic acid ...)copy SMILEScopy InChI
Affinity DataIC50: 281nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61QBTPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents of the University of Minnesota

US Patent
LigandPNGBDBM214699(US9296728, 22)copy SMILEScopy InChI
Affinity DataIC50: 299nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KH0M5RUS Patent
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