Compile Data Set for Download or QSAR
Found 71 of ic50 data for polymerid = 9642
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582891(CHEMBL5078908)copy SMILES
Affinity DataIC50: 3nMAssay Description:Inhibition of SETD2 (unknown origin) preincubated for 30 mins followed by SAM substrate addition measured after 2 hrs by plate reader methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50594410(CHEMBL5178972)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ43XCPubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582889(CHEMBL5073608)copy SMILES
Affinity DataIC50: 7nMAssay Description:Inhibition of SETD2 (unknown origin) preincubated for 30 mins followed by SAM substrate addition measured after 2 hrs by plate reader methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582892(CHEMBL5093241)copy SMILES
Affinity DataIC50: 8nMAssay Description:Inhibition of SETD2 (unknown origin) preincubated for 30 mins followed by SAM substrate addition measured after 2 hrs by plate reader methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582885(CHEMBL5091591)copy SMILES
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582885(CHEMBL5091591)copy SMILES
Affinity DataIC50: 8nMAssay Description:Inhibition of SETD2 (unknown origin) preincubated for 30 mins followed by SAM substrate addition measured after 2 hrs by plate reader methodMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50594410(CHEMBL5178972)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ43XCPubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50594408(CHEMBL5195440)copy SMILES
Affinity DataIC50: 11nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ43XCPubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50594409(CHEMBL5206271)copy SMILES
Affinity DataIC50: 11nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ43XCPubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582878(CHEMBL5082544)copy SMILES
Affinity DataIC50: 12nMAssay Description:Inhibition of SETD2 (unknown origin) preincubated for 30 mins followed by SAM substrate addition measured after 2 hrs by plate reader methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50594403(CHEMBL5189290)copy SMILES
Affinity DataIC50: 12nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ43XCPubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582883(CHEMBL5082960)copy SMILES
Affinity DataIC50: 12nMAssay Description:Inhibition of SETD2 (unknown origin) preincubated for 30 mins followed by SAM substrate addition measured after 2 hrs by plate reader methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582890(CHEMBL5094380)copy SMILES
Affinity DataIC50: 12nMAssay Description:Inhibition of SETD2 (unknown origin) preincubated for 30 mins followed by SAM substrate addition measured after 2 hrs by plate reader methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50594409(CHEMBL5206271)copy SMILES
Affinity DataIC50: 14nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ43XCPubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50594408(CHEMBL5195440)copy SMILES
Affinity DataIC50: 15nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ43XCPubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582880(CHEMBL5071957)copy SMILES
Affinity DataIC50: 15nMAssay Description:Inhibition of SETD2 (unknown origin) preincubated for 30 mins followed by SAM substrate addition measured after 2 hrs by plate reader methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582893(CHEMBL5072597)copy SMILES
Affinity DataIC50: 17nMAssay Description:Inhibition of SETD2 (unknown origin) preincubated for 30 mins followed by SAM substrate addition measured after 2 hrs by plate reader methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582894(CHEMBL5076615)copy SMILES
Affinity DataIC50: 18nMAssay Description:Inhibition of SETD2 (unknown origin) preincubated for 30 mins followed by SAM substrate addition measured after 2 hrs by plate reader methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50594406(EZM-0414 | EZM0414 | Ezm-0414)copy SMILES
Affinity DataIC50: 18nMMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582885(CHEMBL5091591)copy SMILES
Affinity DataIC50: 20nMMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582885(CHEMBL5091591)copy SMILES
Affinity DataIC50: 23nMAssay Description:Inhibition of SETD2 in human A549 cells assessed as H3K36 trimethyl mark incubated for 3 days by in-cell western assayMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582879(CHEMBL5088515)copy SMILES
Affinity DataIC50: 23nMAssay Description:Inhibition of SETD2 (unknown origin) preincubated for 30 mins followed by SAM substrate addition measured after 2 hrs by plate reader methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50594402(CHEMBL5184871)copy SMILES
Affinity DataIC50: 27nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ43XCPubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582889(CHEMBL5073608)copy SMILES
Affinity DataIC50: 29nMAssay Description:Inhibition of SETD2 in human A549 cells assessed as H3K36 trimethyl mark incubated for 3 days by in-cell western assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50594406(EZM-0414 | EZM0414 | Ezm-0414)copy SMILES
Affinity DataIC50: 31nMMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50594403(CHEMBL5189290)copy SMILES
Affinity DataIC50: 41nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ43XCPubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582881(CHEMBL5077994)copy SMILES
Affinity DataIC50: 56nMAssay Description:Inhibition of SETD2 (unknown origin) preincubated for 30 mins followed by SAM substrate addition measured after 2 hrs by plate reader methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582878(CHEMBL5082544)copy SMILES
Affinity DataIC50: 64nMAssay Description:Inhibition of SETD2 in human A549 cells assessed as H3K36 trimethyl mark incubated for 3 days by in-cell western assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582899(CHEMBL5091735)copy SMILES
Affinity DataIC50: 66nMAssay Description:Inhibition of SETD2 (unknown origin) preincubated for 30 mins followed by SAM substrate addition measured after 2 hrs by plate reader methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582880(CHEMBL5071957)copy SMILES
Affinity DataIC50: 74nMAssay Description:Inhibition of SETD2 in human A549 cells assessed as H3K36 trimethyl mark incubated for 3 days by in-cell western assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582890(CHEMBL5094380)copy SMILES
Affinity DataIC50: 93nMAssay Description:Inhibition of SETD2 in human A549 cells assessed as H3K36 trimethyl mark incubated for 3 days by in-cell western assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582903(CHEMBL5071333)copy SMILES
Affinity DataIC50: 101nMAssay Description:Inhibition of SETD2 (unknown origin) preincubated for 30 mins followed by SAM substrate addition measured after 2 hrs by plate reader methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582882(CHEMBL5080149)copy SMILES
Affinity DataIC50: 118nMAssay Description:Inhibition of SETD2 (unknown origin) preincubated for 30 mins followed by SAM substrate addition measured after 2 hrs by plate reader methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582879(CHEMBL5088515)copy SMILES
Affinity DataIC50: 127nMAssay Description:Inhibition of SETD2 in human A549 cells assessed as H3K36 trimethyl mark incubated for 3 days by in-cell western assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50594402(CHEMBL5184871)copy SMILES
Affinity DataIC50: 134nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ43XCPubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582884(CHEMBL5072302)copy SMILES
Affinity DataIC50: 147nMAssay Description:Inhibition of SETD2 (unknown origin) preincubated for 30 mins followed by SAM substrate addition measured after 2 hrs by plate reader methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582881(CHEMBL5077994)copy SMILES
Affinity DataIC50: 162nMAssay Description:Inhibition of SETD2 in human A549 cells assessed as H3K36 trimethyl mark incubated for 3 days by in-cell western assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582891(CHEMBL5078908)copy SMILES
Affinity DataIC50: 175nMAssay Description:Inhibition of SETD2 in human A549 cells assessed as H3K36 trimethyl mark incubated for 3 days by in-cell western assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582894(CHEMBL5076615)copy SMILES
Affinity DataIC50: 235nMAssay Description:Inhibition of SETD2 in human A549 cells assessed as H3K36 trimethyl mark incubated for 3 days by in-cell western assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582883(CHEMBL5082960)copy SMILES
Affinity DataIC50: 257nMAssay Description:Inhibition of SETD2 in human A549 cells assessed as H3K36 trimethyl mark incubated for 3 days by in-cell western assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582882(CHEMBL5080149)copy SMILES
Affinity DataIC50: 340nMAssay Description:Inhibition of SETD2 in human A549 cells assessed as H3K36 trimethyl mark incubated for 3 days by in-cell western assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582893(CHEMBL5072597)copy SMILES
Affinity DataIC50: 379nMAssay Description:Inhibition of SETD2 in human A549 cells assessed as H3K36 trimethyl mark incubated for 3 days by in-cell western assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582892(CHEMBL5093241)copy SMILES
Affinity DataIC50: 384nMAssay Description:Inhibition of SETD2 in human A549 cells assessed as H3K36 trimethyl mark incubated for 3 days by in-cell western assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582903(CHEMBL5071333)copy SMILES
Affinity DataIC50: 397nMAssay Description:Inhibition of SETD2 in human A549 cells assessed as H3K36 trimethyl mark incubated for 3 days by in-cell western assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582884(CHEMBL5072302)copy SMILES
Affinity DataIC50: 449nMAssay Description:Inhibition of SETD2 in human A549 cells assessed as H3K36 trimethyl mark incubated for 3 days by in-cell western assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582899(CHEMBL5091735)copy SMILES
Affinity DataIC50: 540nMAssay Description:Inhibition of SETD2 in human A549 cells assessed as H3K36 trimethyl mark incubated for 3 days by in-cell western assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582901(CHEMBL5085128)copy SMILES
Affinity DataIC50: 674nMAssay Description:Inhibition of SETD2 (unknown origin) preincubated for 30 mins followed by SAM substrate addition measured after 2 hrs by plate reader methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50075101(CHEMBL3414624)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of human SETD2 (1347 to 1711) using histamine H3 (20 to 50) as substrate assessed as transfer of [3H]-Me of [3H-Me]-SAM to peptide substra...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50597882(CHEMBL5187924)copy SMILES
Affinity DataIC50: 800nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DZRPubMed
TargetHistone-lysine N-methyltransferase SETD2(Homo sapiens (Human))TBA
LigandPNGBDBM50582887(CHEMBL5076782)copy SMILES
Affinity DataIC50: 818nMAssay Description:Inhibition of SETD2 (unknown origin) preincubated for 30 mins followed by SAM substrate addition measured after 2 hrs by plate reader methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03D29PubMed
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