TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human ROCK incubated for 20 mins followed by 33P ATP after 120 minsMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of human ROCK incubated for 20 mins followed by 33P ATP after 120 minsMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of ROCK1/2 in human PANC1 cells assessed as reduction in MYPT1 phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Inhibition of ROCK1/2 in human PANC1 cells assessed as reduction in MYPT1 phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 72nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 75nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 75nMAssay Description:Inhibition of ROCK1/2 in human PANC1 cells assessed as reduction in MYPT1 phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 85nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 85nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 87nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 94nMAssay Description:Inhibition of ROCK1/2 in human PANC1 cells assessed as reduction in MYPT1 phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 95nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 116nMAssay Description:Inhibition of ROCK1/2 in human PANC1 cells assessed as reduction in MYPT1 phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 136nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 173nMAssay Description:Inhibition of ROCK1/2 in human PANC1 cells assessed as reduction in MYPT1 phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Universit£ Grenoble Alpes
Curated by ChEMBL
Universit£ Grenoble Alpes
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair