Compile Data Set for Download or QSAR
Found 3 of affinity data with PDB=3EQR
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50246162(CHEMBL472392 | N3-(2,6-dimethylphenyl)-1-(3-methox...)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Inhibition of histidine-tagged ACK1 (amino acids 117 to 489) (unknown origin) expressed in SF9 cellsMore data for this Ligand-Target Pair
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50246162(CHEMBL472392 | N3-(2,6-dimethylphenyl)-1-(3-methox...)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Inhibition of flag-tagged ACK1 (unknown origin) autophosphorylation expressed in human 293 cellsMore data for this Ligand-Target Pair
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50246162(CHEMBL472392 | N3-(2,6-dimethylphenyl)-1-(3-methox...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of ACK1 kinase (unknown origin)More data for this Ligand-Target Pair