TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.00350nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.200nMAssay Description:Agonist activity at human V1B receptor expressed in HEK293 cells assessed as intracellular calcium level measured at 3 secs interval for 5 mins by fu...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.240nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.5nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.800nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 1.5nMAssay Description:Agonist activity at human vasopressin V1b receptor expressed CHO cells assessed as induction of phospholipase C activity after 15 mins by inositol ph...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 1.70nMAssay Description:Binding affinity to human vasopressin V1b receptor expressed CHO cells after 1 hr by spectrofluorimetry analysisMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 2.48nMAssay Description:Agonist activity at human vasopressin V1b receptor expressed CHO cells assessed as induction of phospholipase C activity after 15 mins by inositol ph...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 4.30nMAssay Description:Agonist activity at human vasopressin V1b expressed in HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 4.80nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 6.93nMAssay Description:Agonist activity at human vasopressin V1b receptor expressed CHO cells assessed as induction of phospholipase C activity after 15 mins by inositol ph...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 7.5nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 7.70nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 8nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 8.70nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: >10nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: >10nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: >10nMAssay Description:Agonist activity at human vasopressin V1b expressed in HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: >10nMAssay Description:Agonist activity at human vasopressin V1b expressed in HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: >10nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Antagonism against Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
In DepthDetails
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Agonist activity at human vasopressin V1b expressed in HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Agonist activity at recombinant human V1B receptor expressed in HEK293 cells measured after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 15nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 16nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 18nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 19nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 20nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 21nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 24nMAssay Description:Agonist activity at recombinant human V1B receptor expressed in HEK293 cells measured after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 25nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 26nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 26nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 28nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 28nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 29nMAssay Description:Agonist activity at human V1b receptor expressed in HEK293FT cells incubated for 30 mins by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 29nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 30nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 31nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 32nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 33nMAssay Description:Agonist activity at human vasopressin V1b receptor expressed in CHO cells assessed as increase in intracellular calcium flux measured for 5 mins by F...More data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 37nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 38nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 39nMAssay Description:Agonist activity at human V1b receptor expressed in HEK293FT cells assessed as stimulation of calcium release by Aequorin based assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 39nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 40nMAssay Description:Agonist activity at recombinant human V1B receptor expressed in HEK293 cells measured after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 41nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 44nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 45nMAssay Description:Agonist activity at recombinant human vasopressin V1b receptor expressed in Flp-In-293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University and Department of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 46nMAssay Description:Agonist activity at recombinant human V1B receptor expressed in HEK293 cells measured after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair