TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University of South Carolina Campus
Curated by ChEMBL
Medical University of South Carolina Campus
Curated by ChEMBL
Affinity DataEC50: 54nMAssay Description:Binding affinity to human NTR2 by gamma countingMore data for this Ligand-Target Pair
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University of South Carolina Campus
Curated by ChEMBL
Medical University of South Carolina Campus
Curated by ChEMBL
Affinity DataEC50: 110nMAssay Description:Agonist activity at human NTS2 receptor expressed in HEK293 cells assessed as inhibition of constitutive activity on MAPK-mediated luciferase activit...More data for this Ligand-Target Pair
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University of South Carolina Campus
Curated by ChEMBL
Medical University of South Carolina Campus
Curated by ChEMBL
Affinity DataEC50: 480nMAssay Description:Agonist activity at human NTS2 receptor expressed in HEK293 cells assessed as inhibition of constitutive activity on MAPK-mediated luciferase activit...More data for this Ligand-Target Pair
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University of South Carolina Campus
Curated by ChEMBL
Medical University of South Carolina Campus
Curated by ChEMBL
Affinity DataEC50: 590nMAssay Description:Agonist activity at human NTS2 receptor expressed in HEK293 cells assessed as inhibition of constitutive activity on MAPK-mediated luciferase activit...More data for this Ligand-Target Pair
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University of South Carolina Campus
Curated by ChEMBL
Medical University of South Carolina Campus
Curated by ChEMBL
Affinity DataEC50: 690nMAssay Description:Agonist activity at human NTS2 receptor expressed in HEK293 cells assessed as inhibition of constitutive activity on MAPK-mediated luciferase activit...More data for this Ligand-Target Pair
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University of South Carolina Campus
Curated by ChEMBL
Medical University of South Carolina Campus
Curated by ChEMBL
Affinity DataEC50: 840nMAssay Description:Agonist activity at human NTS2 receptor expressed in HEK293 cells assessed as inhibition of constitutive activity on MAPK-mediated luciferase activit...More data for this Ligand-Target Pair
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University of South Carolina Campus
Curated by ChEMBL
Medical University of South Carolina Campus
Curated by ChEMBL
Affinity DataEC50: >8.00E+4nMAssay Description:Agonist activity at NTR2 in human U2OS cells after 1 hr by beta-arrestin GFP reporter gene assayMore data for this Ligand-Target Pair
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University of South Carolina Campus
Curated by ChEMBL
Medical University of South Carolina Campus
Curated by ChEMBL
Affinity DataEC50: >8.00E+4nMAssay Description:Agonist activity at NTR2 in human U2OS cells after 1 hr by beta-arrestin GFP reporter gene assayMore data for this Ligand-Target Pair