Compile Data Set for Download or QSAR
Found 18 of ec50 data for polymerid = 50006850
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547480(CHEMBL4790235)copy SMILES
Affinity DataEC50:  278nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547479(CHEMBL4794290)copy SMILES
Affinity DataEC50:  393nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547491(CHEMBL4784916)copy SMILES
Affinity DataEC50:  532nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547492(CHEMBL4779693)copy SMILES
Affinity DataEC50:  538nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50078022(CHEMBL3417402)copy SMILEScopy InChI
Affinity DataEC50:  700nMAssay Description:Activation of Bax in human HuH7 cells assessed as inhibition of mitochondrial accumulation of fluorescent probe Mitotracker Red after 12 to 72 hrs by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547481(CHEMBL4777011)copy SMILES
Affinity DataEC50:  704nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547483(CHEMBL4778142)copy SMILES
Affinity DataEC50:  719nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547487(CHEMBL4761391)copy SMILES
Affinity DataEC50:  725nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547484(CHEMBL4780328)copy SMILES
Affinity DataEC50:  809nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547490(CHEMBL4756429)copy SMILES
Affinity DataEC50:  856nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547482(CHEMBL4754714)copy SMILES
Affinity DataEC50:  874nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547489(CHEMBL4758680)copy SMILES
Affinity DataEC50:  925nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547488(CHEMBL4797324)copy SMILES
Affinity DataEC50:  967nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547493(CHEMBL4776616)copy SMILES
Affinity DataEC50:  992nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547485(CHEMBL4753330)copy SMILES
Affinity DataEC50:  1.14E+3nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547486(CHEMBL4790418)copy SMILES
Affinity DataEC50:  2.22E+3nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50078015(CHEMBL3417395)copy SMILEScopy InChI
Affinity DataEC50:  8.20E+3nMAssay Description:Activation of Bax in human HuH7 cells assessed as inhibition of mitochondrial accumulation of fluorescent probe Mitotracker Red after 12 to 72 hrs by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+4nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed