Compile Data Set for Download or QSAR
Found 4 of ec50 data for polymerid = 9090
TargetKappa-type opioid receptor [Y312A](Homo sapiens (Human))
University of North Carolina School of Medicine

LigandPNGBDBM50159165((2S,4aR,6aR,7R,9S,10aS,10bR)-9-(acetyloxy)-2-(fura...)copy SMILEScopy InChI
Affinity DataEC50:  6.20nMpH: 7.4Assay Description:HEK293T cells were co-transfected with plasmids encoding the cAMP biosensor GloSensor-22F (Promega) and the different human KOR variants as described...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P849RPPubMed
TargetKappa-type opioid receptor [Y312A](Homo sapiens (Human))
University of North Carolina School of Medicine

LigandPNGBDBM214798(Dynorphin A (1-17) | YGGFLRRIRPKLK)copy SMILEScopy InChI
Affinity DataEC50:  47nMpH: 7.4Assay Description:HEK293T cells were co-transfected with plasmids encoding the cAMP biosensor GloSensor-22F (Promega) and the different human KOR variants as described...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P849RPPubMed
TargetKappa-type opioid receptor [Y312A](Homo sapiens (Human))
University of North Carolina School of Medicine

LigandPNGBDBM21130(N-methyl-2-phenyl-N-[(5R,7S,8S)-7-(pyrrolidin-1-yl...)copy SMILEScopy InChI
Affinity DataEC50:  65nMpH: 7.4Assay Description:HEK293T cells were co-transfected with plasmids encoding the cAMP biosensor GloSensor-22F (Promega) and the different human KOR variants as described...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P849RPPubMed
TargetKappa-type opioid receptor [Y312A](Homo sapiens (Human))
University of North Carolina School of Medicine

LigandPNGBDBM214799(1xx)copy SMILEScopy InChI
Affinity DataEC50:  360nMpH: 7.4Assay Description:HEK293T cells were co-transfected with plasmids encoding the cAMP biosensor GloSensor-22F (Promega) and the different human KOR variants as described...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P849RPPubMed