Compile Data Set for Download or QSAR
Found 183 of ec50 data for polymerid = 9126
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50019646(2-(alpha-(2,6-Dichlorophenoxy)ethyl)2-imidazoline ...)copy SMILEScopy InChI
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human adrenoceptor aplha 2C expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9ZKTPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50419878(CHEMBL1956195)copy SMILEScopy InChI
Affinity DataEC50:  2nMAssay Description:Agonist activity at human adrenoceptor aplha 2C expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9ZKTPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50420342(CHEMBL2089156)copy SMILEScopy InChI
Affinity DataEC50:  2nMAssay Description:Agonist activity at human alpha2C ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50419878(CHEMBL1956195)copy SMILEScopy InChI
Affinity DataEC50:  2nMAssay Description:Agonist activity at human alpha2C ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50473226(CHEMBL297827)copy SMILEScopy InChI
Affinity DataEC50:  2nMAssay Description:Alpha2c receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D221C4PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50419878(CHEMBL1956195)copy SMILEScopy InChI
Affinity DataEC50:  2nMAssay Description:Agonist activity at human alpha2C adrenoreceptor expressed in CHO cells assessed as extracellular acidification measured after 4 mins by cytosensor m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3FK6PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50420342(CHEMBL2089156)copy SMILEScopy InChI
Affinity DataEC50:  2nMAssay Description:Agonist activity at human alpha2C adrenoreceptor expressed in CHO cells assessed as extracellular acidification measured after 4 mins by cytosensor m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3FK6PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50212995(CHEMBL75030)copy SMILEScopy InChI
Affinity DataEC50:  2.20nMAssay Description:Agonistic activity towards human Alpha-2C adrenergic receptor was measured as ability to inhibit forskolin-stimulated synthesis of cyclic adenosine m...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ70ZD
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50473665(CHEMBL70751)copy SMILEScopy InChI
Affinity DataEC50:  2.80nMAssay Description:Agonist potency at Alpha-2C adrenergic receptor assayed in CHO cells expressing human Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4TCQPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM34572(BRIMONIDINE | CHEMBL844 | MLS000069370 | SMR000058...)copy SMILEScopy InChI
Affinity DataEC50:  3.40nMAssay Description:Effective concentration at Alpha-2C adrenergic receptor from CHO-C4 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0MSTPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50473228(AGN-190837 | CHEMBL297752)copy SMILEScopy InChI
Affinity DataEC50:  4.10nMAssay Description:Alpha-2C adrenergic receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D221C4PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50212997(CHEMBL310335)copy SMILEScopy InChI
Affinity DataEC50:  4.10nMAssay Description:Agonistic activity towards human Alpha-2C adrenergic receptor was measured as ability to inhibit forskolin-stimulated synthesis of cyclic adenosine m...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ70ZD
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50421580(CHEMBL117248)copy SMILEScopy InChI
Affinity DataEC50:  5.60nMAssay Description:Agonist potency at Alpha-2C adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4TCQPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50473672(CHEMBL72768)copy SMILEScopy InChI
Affinity DataEC50:  5.60nMAssay Description:Agonist potency at Alpha-2C adrenergic receptor assayed in CHO cells expressing human Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4TCQPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50417349(CHEMBL1276248)copy SMILEScopy InChI
Affinity DataEC50:  6.30nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B32JFPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50055832((1H-Imidazol-2-yl)-(5-methyl-2,3-dihydro-benzo[1,4...)copy SMILEScopy InChI
Affinity DataEC50:  6.60nMAssay Description:Effective concentration at Alpha-2C adrenergic receptor from CHO-C4 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0MSTPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50473683(CHEMBL72724)copy SMILEScopy InChI
Affinity DataEC50:  7.90nMAssay Description:Agonist potency at Alpha-2C adrenergic receptor assayed in CHO cells expressing human Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4TCQPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50473677(CHEMBL72441)copy SMILEScopy InChI
Affinity DataEC50:  8.90nMAssay Description:Agonist potency at Alpha-2C adrenergic receptor assayed in CHO cells expressing human Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4TCQPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM34572(BRIMONIDINE | CHEMBL844 | MLS000069370 | SMR000058...)copy SMILEScopy InChI
Affinity DataEC50:  9.5nMAssay Description:Alpha-2C adrenergic receptor agonistic potency as inhibition of forskolin-stimulated cyclic adenosine monophosphate synthesisMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DV1N3J
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50218115((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...)copy SMILEScopy InChI
Affinity DataEC50:  10nMAssay Description:Agonistic potency at human adrenergic alpha2C receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W095NPPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50419874(CHEMBL1956192)copy SMILEScopy InChI
Affinity DataEC50:  10nMAssay Description:Agonist activity at human alpha2C ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50218115((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...)copy SMILEScopy InChI
Affinity DataEC50:  10nMAssay Description:Agonistic potency at human adrenergic alpha2C receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W095NPPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50412244(CHEMBL495096)copy SMILEScopy InChI
Affinity DataEC50:  10nMAssay Description:Agonist activity at human recombinant adrenergic Alpha-2C receptor expressed in CHO cells assessed as stimulation of extracellular acidificationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ4147PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50419874(CHEMBL1956192)copy SMILEScopy InChI
Affinity DataEC50:  10nMAssay Description:Agonist activity at human adrenoceptor aplha 2C expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9ZKTPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50218115((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...)copy SMILEScopy InChI
Affinity DataEC50:  10nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B32JFPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50052880(CHEMBL49137 | Imidazolidin-2-ylidene-(5-methyl-qui...)copy SMILEScopy InChI
Affinity DataEC50:  14nMAssay Description:Alpha-2C adrenergic receptor agonistic potency as inhibition of forskolin-stimulated cyclic adenosine monophosphate synthesisMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DV1N3J
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50473229(CHEMBL295186)copy SMILEScopy InChI
Affinity DataEC50:  14nMAssay Description:Alpha2c receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D221C4PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50473669(CHEMBL70692)copy SMILEScopy InChI
Affinity DataEC50:  16nMAssay Description:Agonist potency at Alpha-2C adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4TCQPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50417354(CHEMBL396013)copy SMILEScopy InChI
Affinity DataEC50:  19nMAssay Description:Agonistic potency at human adrenergic alpha2C receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W095NPPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50417354(CHEMBL396013)copy SMILEScopy InChI
Affinity DataEC50:  19nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B32JFPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50412258(CHEMBL451229)copy SMILEScopy InChI
Affinity DataEC50:  21nMAssay Description:Agonist activity at human recombinant adrenergic Alpha-2C receptor expressed in CHO cells assessed as stimulation of extracellular acidificationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ4147PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50473224(CHEMBL296660)copy SMILEScopy InChI
Affinity DataEC50:  21nMAssay Description:Alpha2c receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D221C4PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50193034(CHEMBL3904276)copy SMILEScopy InChI
Affinity DataEC50:  22nMAssay Description:Agonist activity at human alpha2c-AR expressed in CHO cells assessed as rate of acidification after 240 mins by cytosensor microphysiometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2086784PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50493433(CHEMBL2431282)copy SMILEScopy InChI
Affinity DataEC50:  25nMAssay Description:Agonist activity at human alpha2C ARMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50417343(CHEMBL1276140)copy SMILEScopy InChI
Affinity DataEC50:  25nMAssay Description:Agonist activity at human alpha2C ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50212996(CHEMBL306377)copy SMILEScopy InChI
Affinity DataEC50:  25nMAssay Description:Agonistic activity towards human Alpha-2C adrenergic receptor was measured as ability to inhibit forskolin-stimulated synthesis of cyclic adenosine m...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ70ZD
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50417351(CHEMBL1278084)copy SMILEScopy InChI
Affinity DataEC50:  25nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B32JFPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50417343(CHEMBL1276140)copy SMILEScopy InChI
Affinity DataEC50:  25nMAssay Description:Agonist activity at human alpha2C adrenoreceptor expressed in CHO cells assessed as extracellular acidification measured after 4 mins by cytosensor m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3FK6PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50415138(CHEMBL576078)copy SMILEScopy InChI
Affinity DataEC50:  25nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J104DZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50417343(CHEMBL1276140)copy SMILEScopy InChI
Affinity DataEC50:  25nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B32JFPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50473227(CHEMBL50720)copy SMILEScopy InChI
Affinity DataEC50:  27nMAssay Description:Alpha2c receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D221C4PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50473663(CHEMBL553276)copy SMILEScopy InChI
Affinity DataEC50:  28nMAssay Description:Agonist potency at Alpha-2C adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4TCQPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50419889(CHEMBL155866)copy SMILEScopy InChI
Affinity DataEC50:  28nMAssay Description:Agonist activity at human adrenoceptor aplha 2C expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9ZKTPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50473681(CHEMBL540035)copy SMILEScopy InChI
Affinity DataEC50:  28nMAssay Description:Agonist potency at Alpha-2C adrenergic receptor assayed in CHO cells expressing human Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4TCQPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50419884(CHEMBL157955)copy SMILEScopy InChI
Affinity DataEC50:  28nMAssay Description:Agonist activity at human adrenoceptor aplha 2C expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9ZKTPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50213348(CHEMBL72753)copy SMILEScopy InChI
Affinity DataEC50:  31nMAssay Description:Alpha-2C adrenergic receptor agonistic potency as inhibition of forskolin-stimulated cyclic adenosine monophosphate synthesisMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DV1N3J
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50417346(CHEMBL1276220)copy SMILEScopy InChI
Affinity DataEC50:  35nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B32JFPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50417346(CHEMBL1276220)copy SMILEScopy InChI
Affinity DataEC50:  35nMAssay Description:Agonist activity at human alpha2C ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50417344(CHEMBL1276218)copy SMILEScopy InChI
Affinity DataEC50:  40nMAssay Description:Agonist activity at human alpha2C ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50002905(CHEMBL373535)copy SMILEScopy InChI
Affinity DataEC50:  40nMAssay Description:Agonist activity at human adrenergic Alpha-2C receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27Z13PubMed
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