Compile Data Set for Download or QSAR
Found 5 of ic50 data for polymerid = 49000619
TargetGlutamate receptor ionotropic, kainate 3(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50178136((S)-1-(2-amino-2-carboxyethyl)-3-(2-carboxybenzyl)...)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonist activity at recombinant GluK3 receptor (unknown origin) expressed in Xenopus oocyte assessed as inhibition of glutamate-induced current am...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1T0NPubMed
TargetGlutamate receptor ionotropic, kainate 3(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50207594(2,3-Dihydroxy-6-nitro-benzo[f]quinoxaline-7-sulfon...)copy SMILEScopy InChI
Affinity DataIC50: 4.40E+4nMAssay Description:Displacement of [3H]kainate from human GLUK7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69KCTPubMed
TargetGlutamate receptor ionotropic, kainate 3(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50364074(CHEMBL1950805)copy SMILEScopy InChI
Affinity DataIC50: 8.13E+4nMAssay Description:Antagonist activity at human recombinant GluK3 receptor expressed in human HEK293 cells assessed as inhibition of glutamate-stimulated calcium influx...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9XTJPubMed
TargetGlutamate receptor ionotropic, kainate 3(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50185318((S)-1-(2-amino-2-carboxyethyl)-3-(2-carboxythiophe...)copy SMILEScopy InChI
Affinity DataIC50: 2.64E+5nMAssay Description:Displacement of [3H]kainate from human GLUK7 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FQ9W76PubMed
TargetGlutamate receptor ionotropic, kainate 3(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50178148((RS)-1-(2-amino-2-carboxyethyl)-3-(2-carboxybenzyl...)copy SMILEScopy InChI
Affinity DataIC50: 8.80E+5nMAssay Description:Displacement of [3H]kainate from human GLUK7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69KCTPubMed