Compile Data Set for Download or QSAR
Found 467 of ic50 data for polymerid = 50003459,50003477
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517643(CHEMBL4451682)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity in human Raji cell lysates after 1 hr by competitive ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517609(CHEMBL4440581)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity in human Raji cell lysates after 1 hr by competitive ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517607(CHEMBL4590398)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity in human Raji cell lysates after 1 hr by competitive ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517617(CHEMBL4458756)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50230543(CHEMBL5283576)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of human platelet Thromboxane synthetaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC85WVPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517607(CHEMBL4590398)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517643(CHEMBL4451682)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50398608(MARIZOMIB)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of 20S proteasome beta 2c (unknown origin) after 1 hr by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MHBPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517609(CHEMBL4440581)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50426994(CHEMBL2326533)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4DRMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517647(CHEMBL4463326)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50430961(CHEMBL2337844)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of trypsin-like activity of human constitutive 20s proteasome beta-2 subunit using Boc-LRR-AMC as substrate assessed as remaining activity...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F19135PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517633(CHEMBL4471150)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50307481((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of catalytic activity of immunoproteasome 20s subunit beta2 in human Raji cells incubated for 1 hr by BODIPY(FL)-LU-112 probe based compet...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60SJ2PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50307481((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of catalytic activity of immunoproteasome 20s subunit beta2 in human Raji cells incubated for 1 hr by BODIPY(FL)-LU-112 probe based compet...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60SJ2PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50426994(CHEMBL2326533)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity in human Raji cell lysates after 1 hr by competitive ABPP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50430968(CHEMBL2337847)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of trypsin-like activity of human constitutive 20s proteasome beta-2 subunit using Boc-LRR-AMC as substrate assessed as remaining activity...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F19135PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50430969(CHEMBL2337846)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of trypsin-like activity of human constitutive 20s proteasome beta-2 subunit using Boc-LRR-AMC as substrate assessed as remaining activity...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F19135PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517625(CHEMBL4515041)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50430970(CHEMBL2337845)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of trypsin-like activity of human constitutive 20s proteasome beta-2 subunit using Boc-LRR-AMC as substrate assessed as remaining activity...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F19135PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517624(CHEMBL4444586)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517616(CHEMBL4550571)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517596(CHEMBL4450505)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50430962(CHEMBL2337843)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of trypsin-like activity of human constitutive 20s proteasome beta-2 subunit using Boc-LRR-AMC as substrate assessed as remaining activity...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F19135PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50185156(CHEMBL210439 | Hmb-Val-Gln-Leu-VE)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of trypsin like activity of proteasomeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3G5JPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517635(CHEMBL4542603)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50426996(CHEMBL2326261)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of trypsin-like activity of proteasome beta 2 subunit in HEK-293T cell lysates using BODIPY-BODIPY-TMR-epoxomicin as probe after 1 hr by S...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ62VMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517648(CHEMBL4471154)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517618(CHEMBL4546121)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50398608(MARIZOMIB)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Reversible inhibition of human erythrocyte derived 20S proteasome subunit beta2 after 30 mins by fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2668FBFPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50526811(Kzr-616)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Inhibition of 20S proteasome beta 2c (unknown origin) after 1 hr by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MHBPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517613(CHEMBL4549724)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50536425(CHEMBL4563298)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Inhibition of catalytic activity of immunoproteasome 20s subunit beta2 in human Raji cells incubated for 1 hr by BODIPY(FL)-LU-112 probe based compet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60SJ2PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50536425(CHEMBL4563298)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Inhibition of catalytic activity of immunoproteasome 20s subunit beta2 in human Raji cells incubated for 1 hr by BODIPY(FL)-LU-112 probe based compet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60SJ2PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50398609(CHEMBL2141296 | IXAZOMIB CITRATE | Ixazomib | MLN2...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of 20S proteasome beta 2c (unknown origin) after 1 hr by fluorescence based assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517602(CHEMBL4435519)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517649(CHEMBL4457630)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50185159(CHEMBL208162 | Hmb-Phe-Gln-Leu-VE)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of trypsin like activity of proteasomeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3G5JPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517598(CHEMBL4543211)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517623(CHEMBL4467279)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517646(CHEMBL4446148)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517638(CHEMBL4465228)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50185155(CHEMBL207774 | H-Phe-Val-Gln-Leu-VE)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Inhibition of trypsin like activity of proteasomeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3G5JPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517597(CHEMBL4589564)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity (unknown origin) by cell based ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50536438(CHEMBL4534488)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of catalytic activity of immunoproteasome 20s subunit beta2 in human Raji cells incubated for 1 hr by BODIPY(FL)-LU-112 probe based compet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60SJ2PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50536438(CHEMBL4534488)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of catalytic activity of immunoproteasome 20s subunit beta2 in human Raji cells incubated for 1 hr by BODIPY(FL)-LU-112 probe based compet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60SJ2PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50536431(CHEMBL4519899)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of catalytic activity of immunoproteasome 20s subunit beta2 in human Raji cells incubated for 1 hr by BODIPY(FL)-LU-112 probe based compet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60SJ2PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50536438(CHEMBL4534488)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Inhibition of catalytic activity of constitutive proteasome 20s subunit beta2 in human Raji cells incubated for 1 hr by BODIPY(FL)-LU-112 probe based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60SJ2PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50536438(CHEMBL4534488)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Inhibition of catalytic activity of constitutive proteasome 20s subunit beta2 in human Raji cells incubated for 1 hr by BODIPY(FL)-LU-112 probe based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60SJ2PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre

Curated by ChEMBL
LigandPNGBDBM50517618(CHEMBL4546121)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Inhibition of 20S constitutive proteasome beta 2 trypsin-like activity in human Raji cell lysates after 1 hr by competitive ABPP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63XMPubMed
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