Compile Data Set for Download or QSAR
Found 21 of ic50 data for polymerid = 50004512
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371227(CHEMBL400462)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa ExsA binding to DNAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69KD8PubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50319090((E)-3-(4-Acetyl-phenyl)-N-[4-(1-hydroxy-6-nitro-1H...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa 388 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PJ2PubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50378357(CHEMBL575329)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa ExsA binding to DNAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD12KZPubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50319080((E)-N-(4-(6-cyano-1-hydroxy-1H-benzo[d]imidazol-2-...)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PJ2PubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50319088((E)-2-(2-(4-(3-(4-acetylphenyl)acrylamido)phenyl)-...)copy SMILEScopy InChI
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PJ2PubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50371226(CHEMBL251209)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa ExsA binding to DNAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69KD8PubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50319089((E)-2-(2-(4-(3-(6-acetylpyridin-3-yl)acrylamido)ph...)copy SMILEScopy InChI
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PJ2PubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50378358(CHEMBL572948)copy SMILEScopy InChI
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa ExsA binding to DNAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD12KZPubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50378359(CHEMBL575963)copy SMILEScopy InChI
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa ExsA binding to DNAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD12KZPubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50319081((E)-N-(4-(1-hydroxy-6-nitro-1H-benzo[d]imidazol-2-...)copy SMILEScopy InChI
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PJ2PubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50319079((E)-N-(4-(1-hydroxy-6-nitro-1H-benzo[d]imidazol-2-...)copy SMILEScopy InChI
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PJ2PubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50319078((E)-N-(4-(6-cyano-1-hydroxy-1H-benzo[d]imidazol-2-...)copy SMILEScopy InChI
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PJ2PubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50319092((E)-3-(6-acetylpyridin-3-yl)-N-(4-(1-hydroxy-6-nit...)copy SMILEScopy InChI
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa 388 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PJ2PubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50319093((E)-N-(4-(1-hydroxy-6-nitro-1H-benzo[d]imidazol-2-...)copy SMILEScopy InChI
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PJ2PubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50319091((E)-3-(4-acetylphenyl)-N-(4-(6-cyano-1-hydroxy-1H-...)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa 388 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PJ2PubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50319082((E)-3-(6-(1H-imidazol-1-yl)pyridin-3-yl)-N-(4-(1-h...)copy SMILEScopy InChI
Affinity DataIC50: 3.12E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PJ2PubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50319085((E)-3-(4-acetylphenyl)-N-(2-amino-2-oxoethyl)-N-(4...)copy SMILEScopy InChI
Affinity DataIC50: 4.75E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PJ2PubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50319086((E)-3-(4-acetylphenyl)-N-(2-amino-2-oxoethyl)-N-(4...)copy SMILEScopy InChI
Affinity DataIC50: 4.90E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PJ2PubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50319087((E)-2-(3-(4-acetylphenyl)-N-(4-(6-cyano-1-hydroxy-...)copy SMILEScopy InChI
Affinity DataIC50: 5.10E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PJ2PubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50319083((E)-3-(6-(dimethylamino)pyridin-3-yl)-N-(4-(1-hydr...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PJ2PubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50319084((E)-N-(4-(1-hydroxy-6-nitro-1H-benzo[d]imidazol-2-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PJ2PubMed