Compile Data Set for Download or QSAR
Found 88 of ic50 data for polymerid = 50004844
LigandPNGBDBM289504(1-(4-(6-amino-5-(tri- fluoromethyl)pyridin-3- yl)-...)copy SMILEScopy InChI
Ligand InfoPC cidPC sid
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LigandPNGBDBM50609715(CHEMBL5286166)copy SMILES
Ligand Info
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LigandPNGBDBM50609716(CHEMBL5272522)copy SMILES
Ligand Info
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LigandPNGBDBM50609718(CHEMBL5288706)copy SMILES
Ligand Info
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LigandPNGBDBM50609719(CHEMBL5283101)copy SMILES
Ligand Info
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LigandPNGBDBM50609708(CHEMBL5281494)copy SMILES
Ligand InfoPDB
LigandPNGBDBM50609705(CHEMBL5268969)copy SMILES
Ligand Info
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LigandPNGBDBM50609700(CHEMBL5271972)copy SMILES
Ligand Info
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LigandPNGBDBM50609717(CHEMBL5271665)copy SMILES
Ligand Info
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LigandPNGBDBM50609697(GDC-0134 | Gdc-0134 | Rg-6000)copy SMILES
Affinity DataIC50: 11nMMore data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50609714(CHEMBL5270353)copy SMILES
Affinity DataIC50: 12nMMore data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50609712(CHEMBL5276415)copy SMILES
Affinity DataIC50: 13nMMore data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50609710(CHEMBL5276337)copy SMILES
Affinity DataIC50: 13nMMore data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50609711(CHEMBL5268950)copy SMILES
Affinity DataIC50: 13nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM50609701(CHEMBL5277276)copy SMILES
Affinity DataIC50: 14nMMore data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50609707(CHEMBL5284890)copy SMILES
Affinity DataIC50: 17nMMore data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 18.4nMAssay Description:Inhibition of human DLK using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5KB8PubMed
LigandPNGBDBM50609704(CHEMBL5278185)copy SMILES
Affinity DataIC50: 24nMMore data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50609703(CHEMBL5269484)copy SMILES
Affinity DataIC50: 28nMMore data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50059190(CHEMBL3393333)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
LigandPNGBDBM50609702(CHEMBL5278476)copy SMILES
Affinity DataIC50: 47nMMore data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50609699(CHEMBL5284496)copy SMILES
Affinity DataIC50: 53nMMore data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50609709(CHEMBL5273015)copy SMILES
Affinity DataIC50: 53nMMore data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50059191(CHEMBL3393334)copy SMILEScopy InChI
Affinity DataIC50: 57nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
LigandPNGBDBM50609713(CHEMBL5269792)copy SMILES
Affinity DataIC50: 61nMMore data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50059198(CHEMBL3393340)copy SMILEScopy InChI
Affinity DataIC50: 62nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
LigandPNGBDBM50059194(CHEMBL3393337)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
LigandPNGBDBM50059202(CHEMBL3393327)copy SMILEScopy InChI
Affinity DataIC50: 69nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
LigandPNGBDBM50059201(CHEMBL3393329)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
LigandPNGBDBM50609706(CHEMBL5277751)copy SMILES
Affinity DataIC50: 77nMMore data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50059200(CHEMBL3393330)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
LigandPNGBDBM50271208(CHEMBL4128619)copy SMILEScopy InChI
Affinity DataIC50: 99nMAssay Description:Inhibition of doxycycline inducible human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-bas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2639S7KPubMed
LigandPNGBDBM50059207(CHEMBL3393320)copy SMILEScopy InChI
Affinity DataIC50: 109nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
LigandPNGBDBM50059189(CHEMBL3393332)copy SMILEScopy InChI
Affinity DataIC50: 125nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
LigandPNGBDBM50271207(CHEMBL3719135)copy SMILEScopy InChI
Affinity DataIC50: 129nMAssay Description:Inhibition of doxycycline inducible human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs in presence of 10% bovine ser...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2639S7KPubMed
LigandPNGBDBM50059193(CHEMBL3393336)copy SMILEScopy InChI
Affinity DataIC50: 141nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
LigandPNGBDBM50271212(CHEMBL3715238)copy SMILEScopy InChI
Affinity DataIC50: 144nMAssay Description:Inhibition of doxycycline inducible human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-bas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2639S7KPubMed
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Inhibition of human DLK using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W380MTPubMed
LigandPNGBDBM50271240(CHEMBL3718522)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Inhibition of doxycycline inducible human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-bas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2639S7KPubMed
LigandPNGBDBM50059199(CHEMBL3393331)copy SMILEScopy InChI
Affinity DataIC50: 193nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
LigandPNGBDBM50271207(CHEMBL3719135)copy SMILEScopy InChI
Affinity DataIC50: 195nMAssay Description:Inhibition of doxycycline inducible human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-bas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2639S7KPubMed
LigandPNGBDBM50609698(CHEMBL5281886)copy SMILES
Affinity DataIC50: 201nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM50271211(CHEMBL4128477)copy SMILEScopy InChI
Affinity DataIC50: 202nMAssay Description:Inhibition of doxycycline inducible human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-bas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2639S7KPubMed
LigandPNGBDBM50271228(CHEMBL4128889)copy SMILEScopy InChI
Affinity DataIC50: 208nMAssay Description:Inhibition of doxycycline inducible human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-bas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2639S7KPubMed
LigandPNGBDBM50271210(CHEMBL3714822)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Inhibition of doxycycline inducible human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-bas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2639S7KPubMed
LigandPNGBDBM50059197(CHEMBL3393339)copy SMILEScopy InChI
Affinity DataIC50: 213nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
LigandPNGBDBM50059212(CHEMBL3393312)copy SMILEScopy InChI
Affinity DataIC50: 229nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
LigandPNGBDBM50059192(CHEMBL3393335)copy SMILEScopy InChI
Affinity DataIC50: 233nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed
LigandPNGBDBM50271258(CHEMBL3717481)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of doxycycline inducible human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-bas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2639S7KPubMed
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