Compile Data Set for Download or QSAR
Found 119 of ic50 data for polymerid = 50006433
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50552663(CHEMBL4746871)copy SMILES
Affinity DataIC50: 1.69E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged 53BP1 TTD (1484 to1603 residues) expressed in Escherichia coli BL21 (DE3) cells using Biotin-H...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55S4RPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440606(CHEMBL2426376)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50552664(CHEMBL4740162)copy SMILES
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged 53BP1 TTD (1484 to1603 residues) expressed in Escherichia coli BL21 (DE3) cells using Biotin-H...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55S4RPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440602(CHEMBL2426479)copy SMILEScopy InChI
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440599(CHEMBL2426482)copy SMILEScopy InChI
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440601(CHEMBL2426480)copy SMILEScopy InChI
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440613(CHEMBL2426365)copy SMILEScopy InChI
Affinity DataIC50: 8.70E+3nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440604(CHEMBL2426497)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440603(CHEMBL2426498)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440605(CHEMBL2424677)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440607(CHEMBL2426375)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440608(CHEMBL2426374)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440609(CHEMBL2426373)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440610(CHEMBL2426368)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440611(CHEMBL2426367)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440612(CHEMBL2426366)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440614(CHEMBL2426364)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440560(CHEMBL2426363)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440561(CHEMBL2426362)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440562(CHEMBL2426361)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50341828(3-bromo-5-[(4-pyrrolidin-1-ylpiperidin-1-yl)carbon...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440564(CHEMBL2426359)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440565(CHEMBL2426358)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440566(CHEMBL2426478)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440567(CHEMBL2426477)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440568(CHEMBL2426476)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440569(CHEMBL2424678)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440570(CHEMBL2426475)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440571(CHEMBL2426474)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440572(CHEMBL2426473)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440573(CHEMBL2426472)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440574(CHEMBL2426471)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440575(CHEMBL2426470)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440576(CHEMBL2426469)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440577(CHEMBL2426468)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440578(CHEMBL2426467)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440579(CHEMBL2426466)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440580(CHEMBL2426465)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440581(CHEMBL2426464)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440582(CHEMBL2426463)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440583(CHEMBL2426462)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440584(CHEMBL2426461)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440585(CHEMBL2426496)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440586(CHEMBL2426495)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440587(CHEMBL2426494)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440588(CHEMBL2426493)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440589(CHEMBL2426492)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440590(CHEMBL2426491)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440591(CHEMBL2426490)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetTP53-binding protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50440592(CHEMBL2426489)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 53BP1 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
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