Compile Data Set for Download or QSAR
Found 312 of ic50 data for polymerid = 9153
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396227(6-[5-Bromo-6-(2-oxa-6-aza-spiro[3.3]hept-6-yl)-pyr...)copy SMILEScopy InChI
Affinity DataIC50: 0.0200nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396236(6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 0.0200nMAssay Description:Inhibition of human GOAT expressed in HEK293 cells harboring -preproghrelin in presence of Octanoate-BSA incubated for 5 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6W53PubMed
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396236(6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 0.0200nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396194(6-(5-Bromo-6-methoxy-pyridin-2-ylmethyl)-5-methyl-...)copy SMILEScopy InChI
Affinity DataIC50: 0.0220nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396205(6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 0.0260nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396220(6-(5-Bromo-6-morpholin-4-yl-pyridin-2-ylmethyl)-5-...)copy SMILEScopy InChI
Affinity DataIC50: 0.0260nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396246(6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 0.0270nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396239(6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 0.0270nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50548078(CHEMBL4746798)copy SMILES
Affinity DataIC50: 0.0280nMAssay Description:Inhibition of human GOAT expressed in HEK293 cells harboring -preproghrelin in presence of Octanoate-BSA incubated for 5 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6W53PubMed
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396118(6-(5,6-Dibromo-pyridin-2-ylmethyl)-5-methyl-[1,2,5...)copy SMILEScopy InChI
Affinity DataIC50: 0.0300nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396219(1-[6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyr...)copy SMILEScopy InChI
Affinity DataIC50: 0.0330nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396233(6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 0.0330nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396197(6-[5-Bromo-6-(2-fluoro-ethoxy)-pyridin-2-ylmethyl]...)copy SMILEScopy InChI
Affinity DataIC50: 0.0340nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396112(6-(6-Bromo-5-difluoromethoxy-pyridin-2-ylmethyl)-5...)copy SMILEScopy InChI
Affinity DataIC50: 0.0380nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396222(6-(5-Bromo-6-cyclopropylamino-pyridin-2-ylmethyl)-...)copy SMILEScopy InChI
Affinity DataIC50: 0.0380nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396218(6-{5-Bromo-6-[(3-methyl-oxetan-3-ylmethyl)-amino]-...)copy SMILEScopy InChI
Affinity DataIC50: 0.0450nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396240(6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 0.0460nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396116(6-(5-Brom32.2-chloro-pyridin-2-ylmethyl)-5-methyl-...)copy SMILEScopy InChI
Affinity DataIC50: 0.0470nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396164(6-(6-Amino-5-thiazol-5-yl-pyridin-2-ylmethyl)-5-me...)copy SMILEScopy InChI
Affinity DataIC50: 0.0500nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396226(6-[5-Bromo-6-(3,3-difluoro-azetidin-1-yl)-pyridin-...)copy SMILEScopy InChI
Affinity DataIC50: 0.0520nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396234(6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 0.0540nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396241(6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 0.0550nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396221(3-[6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyr...)copy SMILEScopy InChI
Affinity DataIC50: 0.0560nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396189(6-[5-Bromo-6-(2,2-difluoro-ethoxy)-pyridin-2-yl me...)copy SMILEScopy InChI
Affinity DataIC50: 0.0580nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396191(1-[6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyr...)copy SMILEScopy InChI
Affinity DataIC50: 0.0580nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396119(6-(5-Brom32.2-fluoro-pyridin-2-ylmethyl)-5-methyl-...)copy SMILEScopy InChI
Affinity DataIC50: 0.0660nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50548079(CHEMBL4754865)copy SMILES
Affinity DataIC50: 0.0660nMAssay Description:Inhibition of human GOAT expressed in HEK293 cells harboring -preproghrelin in presence of Octanoate-BSA incubated for 5 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6W53PubMed
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396196(6-[5-Bromo-6-(2,2-difluoro-propoxy)-pyridin-2-ylme...)copy SMILEScopy InChI
Affinity DataIC50: 0.0720nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396139(6-(7-amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 0.0730nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396198(6-[5-Bromo-6-(3-fluoro-propoxy)-pyridin-2-yl methy...)copy SMILEScopy InChI
Affinity DataIC50: 0.0740nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396199(6-(5-Bromo-6-methylsulfanyl-pyridin-2-ylmethyl)-5-...)copy SMILEScopy InChI
Affinity DataIC50: 0.0740nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396235(6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 0.0750nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396180(6-[5-bromo-4-(trifluoromethyl)pyrimidin-2-yl]methy...)copy SMILEScopy InChI
Affinity DataIC50: 0.0770nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396193(6-[5-Bromo-6-(2,2,2-trifluoro-ethoxy)-pyridin-2-yl...)copy SMILEScopy InChI
Affinity DataIC50: 0.0790nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396192(6-[5-Bromo-6-(3-methyl-oxetan-3-ylmethoxy)-pyridin...)copy SMILEScopy InChI
Affinity DataIC50: 0.0820nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396120(6-(5-Brom32.2-difluoromethoxy-pyridin-2-ylmethyl)-...)copy SMILEScopy InChI
Affinity DataIC50: 0.0820nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396167(6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 0.0820nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396215(6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 0.0850nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396200(6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 0.0860nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396216(6-(6-Amino-5-difluoromethoxy-pyridin-2-ylmethyl)-5...)copy SMILEScopy InChI
Affinity DataIC50: 0.0910nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396206(6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 0.0930nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396225(6-[5-Bromo-6-(3,3-difluoro-cyclobutylamino)-pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 0.0960nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396228(1-[6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyr...)copy SMILEScopy InChI
Affinity DataIC50: 0.0970nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396230(6-[5-Bromo-6-(3,3-difluoro-propylamino)-pyridin-2-...)copy SMILEScopy InChI
Affinity DataIC50: 0.0990nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396208(6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396224(3-[6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyr...)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396161(1-[6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyr...)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396224(3-[6-(7-Amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyr...)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396154(6-(6-Furan-2-yl-pyridin-2-ylmethyl)-5-methyl-[1,2,...)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396229(6-[5-Bromo-6-(3,3-difluoro-pyrrolidin-1-yl)-pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Cells are plated with a density of 5000 cells/well in 384-well poly-D-lysin plates and incubated for 1 day at 37° C., 5% CO2 in DMEM medium, 10% FCS,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VH5R5SUS Patent
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