Compile Data Set for Download or QSAR
Found 320 of ki data for polymerid = 1810,50000181
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50246899((S)-2-(3-((S)-1-carboxy-5-(4-iodobenzamido)pentyl)...)copy SMILEScopy InChI
Affinity DataKi:  0.00300nMAssay Description:Inhibition of antiTEV-tagged GCP2 extracellular portion (aa 44-750) (unknown origin) using folyl-di-L-glutamate as substrate by HPLC-based enzymatic ...More data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50089452(CHEMBL3578201)copy SMILEScopy InChI
Affinity DataKi:  0.00860nMAssay Description:Inhibition of antiTEV-tagged GCP2 extracellular portion (aa 44-750) (unknown origin) using folyl-di-L-glutamate as substrate by HPLC-based enzymatic ...More data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50246899((S)-2-(3-((S)-1-carboxy-5-(4-iodobenzamido)pentyl)...)copy SMILEScopy InChI
Affinity DataKi:  0.0100nMAssay Description:Inhibition of GCP2 by top scintillation counter in presence of 30 nM NAA[3]GMore data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50246899((S)-2-(3-((S)-1-carboxy-5-(4-iodobenzamido)pentyl)...)copy SMILEScopy InChI
Affinity DataKi:  0.0100nMAssay Description:Inhibition of PSMA in human LNCaP cell extract using [3H]NAAG by fluorescence-based assayMore data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50246899((S)-2-(3-((S)-1-carboxy-5-(4-iodobenzamido)pentyl)...)copy SMILEScopy InChI
Affinity DataKi:  0.0100nMAssay Description:Inhibition of PSMA in human LNCaP cell extract using [3H]NAAG by radiometric assayMore data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM456924(US10736974, Compound YC-I-27)copy SMILEScopy InChI
Affinity DataKi:  0.0100nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29C71GJUS Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50246899((S)-2-(3-((S)-1-carboxy-5-(4-iodobenzamido)pentyl)...)copy SMILEScopy InChI
Affinity DataKi:  0.0100nMAssay Description:Binding affinity to NAALADaseMore data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50246899((S)-2-(3-((S)-1-carboxy-5-(4-iodobenzamido)pentyl)...)copy SMILEScopy InChI
Affinity DataKi:  0.0100nMAssay Description:Inhibition of PSMA (unknown origin)More data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM456928(US10736974, Compound XY-44)copy SMILEScopy InChI
Affinity DataKi:  0.0170nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29C71GJUS Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50089451(CHEMBL3578202)copy SMILEScopy InChI
Affinity DataKi:  0.0180nMAssay Description:Inhibition of antiTEV-tagged GCP2 extracellular portion (aa 44-750) (unknown origin) using folyl-di-L-glutamate as substrate by HPLC-based enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2X70PubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM456930(US10736974, Compound XY-59)copy SMILEScopy InChI
Affinity DataKi:  0.0200nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29C71GJUS Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM456923(US10736974, Compound DCIBC)copy SMILEScopy InChI
Affinity DataKi:  0.0300nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29C71GJUS Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM578399(US11478558, Compound L9)copy SMILES
Affinity DataKi:  0.0350nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20P138QUS Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM456931(US10736974, Compound XY-58)copy SMILEScopy InChI
Affinity DataKi:  0.0360nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29C71GJUS Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50046832(CHEMBL3309678)copy SMILEScopy InChI
Affinity DataKi:  0.0449nMAssay Description:Inhibition of human recombinant N-terminal Avi-tagged glutamate carboxypeptidase 2 extracellular domain (44 to 750 amino acids) using pteroyl-di-L-gl...More data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50046832(CHEMBL3309678)copy SMILEScopy InChI
Affinity DataKi:  0.0450nMAssay Description:Inhibition of antiTEV-tagged GCP2 extracellular portion (aa 44-750) (unknown origin) using folyl-di-L-glutamate as substrate by HPLC-based enzymatic ...More data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50089454(CHEMBL3578199)copy SMILEScopy InChI
Affinity DataKi:  0.0490nMAssay Description:Inhibition of antiTEV-tagged GCP2 extracellular portion (aa 44-750) (unknown origin) using folyl-di-L-glutamate as substrate by HPLC-based enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2X70PubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM479434(US10894807, ID P242)copy SMILEScopy InChI
Affinity DataKi:  0.0700nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SN0D25US Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50089455(CHEMBL3578197)copy SMILEScopy InChI
Affinity DataKi:  0.0710nMAssay Description:Inhibition of antiTEV-tagged GCP2 extracellular portion (aa 44-750) (unknown origin) using folyl-di-L-glutamate as substrate by HPLC-based enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2X70PubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM642537(US20230414794, Compound S2)copy SMILES
Affinity DataKi:  0.0800nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM456929(US10736974, Compound XY-45)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29C71GJUS Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM17759((2S)-2-(phosphonomethyl)pentanedioic acid | (S)-2-...)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Binding affinity to NAALADaseMore data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50089453(CHEMBL3578200)copy SMILEScopy InChI
Affinity DataKi:  0.110nMAssay Description:Inhibition of antiTEV-tagged GCP2 extracellular portion (aa 44-750) (unknown origin) using folyl-di-L-glutamate as substrate by HPLC-based enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2X70PubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM578398(US11478558, Compound L8)copy SMILES
Affinity DataKi:  0.120nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20P138QUS Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50454862(CHEMBL4211875)copy SMILEScopy InChI
Affinity DataKi:  0.140nMAssay Description:Inhibition of PSMA in human LNCaP cell lysates incubated for 2 hrs in presence of N-acetylaspartylglutamate by Amplex red glutamic acid/glutamate oxi...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN3BGJPubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM479437(US10894807, ID P246)copy SMILEScopy InChI
Affinity DataKi:  0.160nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SN0D25US Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50046850(CHEMBL3311268)copy SMILEScopy InChI
Affinity DataKi:  0.170nMAssay Description:Inhibition of antiTEV-tagged GCP2 extracellular portion (aa 44-750) (unknown origin) using folyl-di-L-glutamate as substrate by HPLC-based enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2X70PubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50046850(CHEMBL3311268)copy SMILEScopy InChI
Affinity DataKi:  0.174nMAssay Description:Inhibition of human recombinant N-terminal Avi-tagged glutamate carboxypeptidase 2 extracellular domain (44 to 750 amino acids) using pteroyl-di-L-gl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NK3GP8PubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50246934((S)-2-(3-((S)-1-carboxy-5-(4-fluorobenzamido)penty...)copy SMILEScopy InChI
Affinity DataKi:  0.194nMAssay Description:Inhibition of PSMA in human LNCaP cell extract using [3H]NAAG by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0NKJPubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM17659((R,S)-2-phosphonomethylpentanedioic acid | 2-(phos...)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:In vitro inhibitory activity against glutamate carboxypeptidase II (GCP II) using N-acetyl-L-aspartyl-[3H]-L-glutamate as a substrateMore data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM17659((R,S)-2-phosphonomethylpentanedioic acid | 2-(phos...)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Concentration of the compound required for the neuroprotective effect determined by inhibition of GCP IIMore data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM479458(US10894807, ID P278)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SN0D25US Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM479453(US10894807, ID P273)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SN0D25US Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM479450(US10894807, ID P270)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SN0D25US Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM479444(US10894807, ID P253)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SN0D25US Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50046831(CHEMBL3309680)copy SMILEScopy InChI
Affinity DataKi:  0.221nMAssay Description:Inhibition of human recombinant N-terminal Avi-tagged glutamate carboxypeptidase 2 extracellular domain (44 to 750 amino acids) using pteroyl-di-L-gl...More data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50246934((S)-2-(3-((S)-1-carboxy-5-(4-fluorobenzamido)penty...)copy SMILEScopy InChI
Affinity DataKi:  0.256nMAssay Description:Inhibition of PSMA in human LNCaP cell extract using [3H]NAAG by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0NKJPubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM456920(US10736974, Entry 23)copy SMILEScopy InChI
Affinity DataKi:  0.260nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29C71GJUS Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM578394(US11478558, Compound L4)copy SMILES
Affinity DataKi:  0.265nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20P138QUS Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM578392(US11478558, Compound L2)copy SMILES
Affinity DataKi:  0.265nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20P138QUS Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50046835(CHEMBL3309676)copy SMILEScopy InChI
Affinity DataKi:  0.268nMAssay Description:Inhibition of human recombinant N-terminal Avi-tagged glutamate carboxypeptidase 2 extracellular domain (44 to 750 amino acids) using pteroyl-di-L-gl...More data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM17659((R,S)-2-phosphonomethylpentanedioic acid | 2-(phos...)copy SMILEScopy InChI
Affinity DataKi:  0.280nMAssay Description:Inhibition of antiTEV-tagged GCP2 extracellular portion (aa 44-750) (unknown origin) using folyl-di-L-glutamate as substrate by HPLC-based enzymatic ...More data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM479415(US10894807, ID P200)copy SMILEScopy InChI
Affinity DataKi: <0.300nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SN0D25US Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM17759((2S)-2-(phosphonomethyl)pentanedioic acid | (S)-2-...)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Inhibition of GCPII (unknown origin) NAALADase activityMore data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM456925(US10736974, Compound YC-I-26)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:The PSMA inhibitory activity was determined using a modification of the fluorescence-based Amplex Red Glutamic Acid Assay. Briefly, lysates of LNCaP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29C71GJUS Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM479431(US10894807, ID P238)copy SMILEScopy InChI
Affinity DataKi: <0.300nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SN0D25US Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM17659((R,S)-2-phosphonomethylpentanedioic acid | 2-(phos...)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Binding affinity to NAALADaseMore data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM479449(US10894807, ID P266)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SN0D25US Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM479429(US10894807, ID P235)copy SMILEScopy InChI
Affinity DataKi: <0.300nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SN0D25US Patent
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Academy of Sciences of the Czech Republic

Curated by ChEMBL
LigandPNGBDBM50046843(CHEMBL3309670)copy SMILEScopy InChI
Affinity DataKi:  0.312nMAssay Description:Inhibition of human recombinant N-terminal Avi-tagged glutamate carboxypeptidase 2 extracellular domain (44 to 750 amino acids) using pteroyl-di-L-gl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NK3GP8PubMed
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