TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Centre de Recherches
Curated by ChEMBL
Centre de Recherches
Curated by ChEMBL
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Centre de Recherches
Curated by ChEMBL
Centre de Recherches
Curated by ChEMBL
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Centre de Recherches
Curated by ChEMBL
Centre de Recherches
Curated by ChEMBL
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Centre de Recherches
Curated by ChEMBL
Centre de Recherches
Curated by ChEMBL
Affinity DataKi: >1.40E+3nMAssay Description:Inhibition of recombinant ERBB2 after 1 hr by scintillation counter analysis in presence of gamma-[33P]ATPMore data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Centre de Recherches
Curated by ChEMBL
Centre de Recherches
Curated by ChEMBL
Affinity DataKi: >1.44E+3nMAssay Description:Inhibition of ERBB2More data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Centre de Recherches
Curated by ChEMBL
Centre de Recherches
Curated by ChEMBL
Affinity DataKi: 3.10E+3nMAssay Description:Inhibition of ERBB2 autophosphorylation Thr 1139 residue in human BT474 cells at 2 to 14 uM after 12 hrs by fluorescence assayMore data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Centre de Recherches
Curated by ChEMBL
Centre de Recherches
Curated by ChEMBL
Affinity DataKi: 3.00E+4nMAssay Description:Binding affinity to ErbB-2More data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Centre de Recherches
Curated by ChEMBL
Centre de Recherches
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of ERBB2More data for this Ligand-Target Pair