Compile Data Set for Download or QSAR
Found 10 of ki data for polymerid = 5620
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))
Pfizer Worldwide R&D

LigandPNGBDBM209866(PF-06651600 | US11111242, Example 5 | US2023034848...)copy SMILES
Affinity DataKi:  32.4nMpH: 7.5Assay Description:Assay buffer was 20 mM HEPES, pH 7.5, 10 mM MgCl2, 0.01% BSA, 1 mM DTT, 0.0005% Tween 20, and 2% DMSO. Inactivation kinetic reactions were performed ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN94F8PubMed
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))
Pfizer Worldwide R&D

LigandPNGBDBM50515526(CHEMBL4452230)copy SMILEScopy InChI
Affinity DataKi:  170nMAssay Description:Inhibition of BLK (unknown origin) using KVEKIGEGTYGVVYK as substrate in presence of [gamma33P]ATP as substrate in presence of [gamma33P]ATP by scint...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85CHNPubMed
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))
Pfizer Worldwide R&D

LigandPNGBDBM50089575(CHEMBL3578214)copy SMILEScopy InChI
Affinity DataKi:  190nMAssay Description:Inhibition of BLK (unknown origin) using KVEKIGEGTYGVVYK as substrate in presence of [gamma33P]ATP as substrate in presence of [gamma33P]ATP by scint...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85CHNPubMed
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))
Pfizer Worldwide R&D

LigandPNGBDBM50402020(CHEMBL2205426)copy SMILEScopy InChI
Affinity DataKi: >1.40E+3nMAssay Description:Inhibition of recombinant BLK after 1 hr by scintillation counter analysis in presence of gamma-[33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8GQ3PubMed
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))
Pfizer Worldwide R&D

LigandPNGBDBM50224883(7-chloro-3-oxo-8-[(thiazol-5-ylmethyl)-amino]-11,1...)copy SMILEScopy InChI
Affinity DataKi: >1.45E+3nMAssay Description:Inhibition of BLKMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X067WTPubMed
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))
Pfizer Worldwide R&D

LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z430BPubMed
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))
Pfizer Worldwide R&D

LigandPNGBDBM50463484(CHEMBL4248525)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of Blk (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC85HXPubMed
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))
Pfizer Worldwide R&D

LigandPNGBDBM50463479(CHEMBL4249925)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of Blk (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC85HXPubMed
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))
Pfizer Worldwide R&D

LigandPNGBDBM50237710(4-methyl-N-[3-(4-methyl-1H-imidazol-1-yl)-5-(trifl...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z430BPubMed
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))
Pfizer Worldwide R&D

LigandPNGBDBM209866(PF-06651600 | US11111242, Example 5 | US2023034848...)copy SMILES
Affinity DataKi:  3.24E+4nMAssay Description:Inhibition of full length recombinant human His-tagged cytoplasmic BLK expressed in baculovirus expression system by KT236 probe based TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3JC2PubMed