Compile Data Set for Download or QSAR
Found 38 of ki data for polymerid = 6339
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190690(US9181233, 67)copy SMILEScopy InChI
Affinity DataKi:  10nM ΔG°:  -46.4kJ/mole IC50: 80nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM124974(US8772508, 8)copy SMILEScopy InChI
Affinity DataKi:  11nM IC50: 580nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R78CW3US Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM50299866(CHEMBL578153 | N-(1-(3-(5-Methyl-1H-imidazol-1-yl)...)copy SMILEScopy InChI
Affinity DataKi:  34nM IC50: 430nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R78CW3US Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190685(US9181233, 60)copy SMILEScopy InChI
Affinity DataKi:  40nM ΔG°:  -42.9kJ/mole IC50: 450nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM50299867(CHEMBL565907 | N-(1-(3-(5-Methyl-1H-imidazol-1-yl)...)copy SMILEScopy InChI
Affinity DataKi:  41nM IC50: 230nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R78CW3US Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190679(US9181233, 52)copy SMILEScopy InChI
Affinity DataKi:  50nM ΔG°:  -42.4kJ/mole IC50: 680nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM50299865(CHEMBL567406 | N-(-1-(3-(5-Methyl-1H-imidazol-1-yl...)copy SMILEScopy InChI
Affinity DataKi:  51nM IC50: 320nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R78CW3US Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM124971(US8772508, 2)copy SMILEScopy InChI
Affinity DataKi:  55nM IC50: 530nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R78CW3US Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190676(US9181233, 47)copy SMILEScopy InChI
Affinity DataKi:  60nM ΔG°:  -41.9kJ/mole IC50: 400nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190680(US9181233, 54)copy SMILEScopy InChI
Affinity DataKi:  60nM ΔG°:  -41.9kJ/mole IC50: 590nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM124975(US8772508, 9)copy SMILEScopy InChI
Affinity DataKi:  67nM IC50: 340nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R78CW3US Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM50299868(CHEMBL565908 | N-(1-(3-(5-Methyl-1H-imidazol-1-yl)...)copy SMILEScopy InChI
Affinity DataKi:  67nM IC50: 460nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R78CW3US Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM124973(US8772508, 4)copy SMILEScopy InChI
Affinity DataKi:  76nM IC50: 730nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R78CW3US Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190695(US9181233, 86)copy SMILEScopy InChI
Affinity DataKi:  80nM ΔG°:  -41.2kJ/mole IC50: 290nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM50299864(CHEMBL574357 | N-(1-(3-(5-Methyl-1H-imidazol-1-yl)...)copy SMILEScopy InChI
Affinity DataKi:  80nM IC50: 340nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R78CW3US Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190687(US9181233, 62)copy SMILEScopy InChI
Affinity DataKi:  80nM ΔG°:  -41.2kJ/mole IC50: 480nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190671(US9181233, 10)copy SMILEScopy InChI
Affinity DataKi:  80nM ΔG°:  -41.2kJ/mole IC50: 480nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190681(US9181233, 55)copy SMILEScopy InChI
Affinity DataKi:  80nM ΔG°:  -41.2kJ/mole IC50: 490nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190678(US9181233, 50)copy SMILEScopy InChI
Affinity DataKi:  80nM ΔG°:  -41.2kJ/mole IC50: 760nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190677(US9181233, 49)copy SMILEScopy InChI
Affinity DataKi:  90nM ΔG°:  -40.9kJ/mole IC50: 360nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM124972(US8772508, 3)copy SMILEScopy InChI
Affinity DataKi:  96nM IC50: 620nMpH: 8.0Assay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30C. QC activity was evaluated fluorometrically...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R78CW3US Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190688(US9181233, 63)copy SMILEScopy InChI
Affinity DataKi:  100nM ΔG°:  -40.6kJ/mole IC50: 220nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190694(US9181233, 85)copy SMILEScopy InChI
Affinity DataKi:  100nM ΔG°:  -40.6kJ/mole IC50: 470nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190669(US9181233, 8)copy SMILEScopy InChI
Affinity DataKi:  110nM ΔG°:  -40.4kJ/mole IC50: 640nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190672(US9181233, 22)copy SMILEScopy InChI
Affinity DataKi:  120nM ΔG°:  -40.2kJ/mole IC50: 520nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190689(US9181233, 65)copy SMILEScopy InChI
Affinity DataKi:  120nM ΔG°:  -40.2kJ/mole IC50: 530nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190696(US9181233, 87)copy SMILEScopy InChI
Affinity DataKi:  120nM ΔG°:  -40.2kJ/mole IC50: 550nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190684(US9181233, 59)copy SMILEScopy InChI
Affinity DataKi:  120nM ΔG°:  -40.2kJ/mole IC50: 560nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190693(US9181233, 84)copy SMILEScopy InChI
Affinity DataKi:  120nM ΔG°:  -40.2kJ/mole IC50: 570nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190674(US9181233, 39)copy SMILEScopy InChI
Affinity DataKi:  130nM ΔG°:  -40.0kJ/mole IC50: 800nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190682(US9181233, 57)copy SMILEScopy InChI
Affinity DataKi:  130nM ΔG°:  -40.0kJ/mole IC50: 830nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190692(US9181233, 83)copy SMILEScopy InChI
Affinity DataKi:  140nM ΔG°:  -39.8kJ/mole IC50: 570nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190683(US9181233, 58)copy SMILEScopy InChI
Affinity DataKi:  140nM ΔG°:  -39.8kJ/mole IC50: 720nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190691(US9181233, 68)copy SMILEScopy InChI
Affinity DataKi:  150nM ΔG°:  -39.6kJ/mole IC50: 410nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190686(US9181233, 61)copy SMILEScopy InChI
Affinity DataKi:  170nM ΔG°:  -39.3kJ/mole IC50: 760nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190675(US9181233, 46)copy SMILEScopy InChI
Affinity DataKi:  180nM ΔG°:  -39.1kJ/mole IC50: 640nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190670(US9181233, 9)copy SMILEScopy InChI
Affinity DataKi:  200nM ΔG°:  -38.9kJ/mole IC50: 760nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent
TargetGlutaminyl-peptide cyclotransferase-like protein(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM190673(US9181233, 24)copy SMILEScopy InChI
Affinity DataKi:  230nM ΔG°:  -38.5kJ/mole IC50: 850nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S46QQHUS Patent