Found 106 hits of Enzyme Inhibition Constant Data
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
DuPont Pharmaceuticals Company
Curated by ChEMBL
DuPont Pharmaceuticals Company
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:In vitro activity against human Plasma kallikrein.More data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
DuPont Pharmaceuticals Company
Curated by ChEMBL
DuPont Pharmaceuticals Company
Curated by ChEMBL
Affinity DataKi: 87nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
DuPont Pharmaceuticals Company
Curated by ChEMBL
DuPont Pharmaceuticals Company
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
DuPont Pharmaceuticals Company
Curated by ChEMBL
DuPont Pharmaceuticals Company
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
DuPont Pharmaceuticals Company
Curated by ChEMBL
DuPont Pharmaceuticals Company
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
DuPont Pharmaceuticals Company
Curated by ChEMBL
DuPont Pharmaceuticals Company
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
DuPont Pharmaceuticals Company
Curated by ChEMBL
DuPont Pharmaceuticals Company
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
DuPont Pharmaceuticals Company
Curated by ChEMBL
DuPont Pharmaceuticals Company
Curated by ChEMBL
Affinity DataKi: 150nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
DuPont Pharmaceuticals Company
Curated by ChEMBL
DuPont Pharmaceuticals Company
Curated by ChEMBL
Affinity DataKi: 220nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
DuPont Pharmaceuticals Company
Curated by ChEMBL
DuPont Pharmaceuticals Company
Curated by ChEMBL
Affinity DataKi: 250nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 360nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 380nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 450nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 480nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 890nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 910nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
DuPont Pharmaceuticals Company
Curated by ChEMBL
DuPont Pharmaceuticals Company
Curated by ChEMBL
Affinity DataKi: >1.60E+3nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Binding affinity against human coagulation factor XMore data for this Ligand-Target Pair
TargetVitamin K-dependent protein C(Homo sapiens (Human))
DuPont Pharmaceuticals Company
Curated by ChEMBL
DuPont Pharmaceuticals Company
Curated by ChEMBL
Affinity DataKi: 1.80E+3nMAssay Description:In vitro activity against human Activated protein CMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+3nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:In vitro activity against human factor IXaMore data for this Ligand-Target Pair
Affinity DataKi: 2.80E+3nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 5.80E+3nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 7.40E+3nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+4nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 1.40E+4nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 1.40E+4nMAssay Description:In vitro activity against human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: >1.50E+4nMAssay Description:The compound was tested for inhibition of human coagulation factor VIIMore data for this Ligand-Target Pair
Affinity DataKi: >1.70E+4nMAssay Description:In vitro activity against human Chymotrypsinogen B1More data for this Ligand-Target Pair
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