Found 60 hits of Enzyme Inhibition Constant Data
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wake Forest University School of Medicine
Curated by ChEMBL
Wake Forest University School of Medicine
Curated by ChEMBL
Affinity DataKi: 2.85E+3nMAssay Description:Binding affinity at dopamine receptor D2 on Sf9 cells by [125I]-IABN displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Wake Forest University School of Medicine
Curated by ChEMBL
Wake Forest University School of Medicine
Curated by ChEMBL
Affinity DataKi: 2.93E+3nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to Sigma opioid receptor of guiena pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Wake Forest University School of Medicine
Curated by ChEMBL
Wake Forest University School of Medicine
Curated by ChEMBL
Affinity DataKi: 3.08E+3nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to Sigma opioid receptor of guiena pig brain membraneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wake Forest University School of Medicine
Curated by ChEMBL
Wake Forest University School of Medicine
Curated by ChEMBL
Affinity DataKi: 3.57E+3nMAssay Description:Binding affinity at dopamine receptor D2 on Sf9 cells by [125I]-IABN displacement.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wake Forest University School of Medicine
Curated by ChEMBL
Wake Forest University School of Medicine
Curated by ChEMBL
Affinity DataKi: 3.60E+3nMAssay Description:Binding affinity at dopamine receptor D2 on Sf9 cells by [125I]-IABN displacement.More data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wake Forest University School of Medicine
Curated by ChEMBL
Wake Forest University School of Medicine
Curated by ChEMBL
Affinity DataKi: 3.76E+3nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]-IABN displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Wake Forest University School of Medicine
Curated by ChEMBL
Wake Forest University School of Medicine
Curated by ChEMBL
Affinity DataKi: 5.48E+3nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to Sigma opioid receptor of guiena pig brain membraneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wake Forest University School of Medicine
Curated by ChEMBL
Wake Forest University School of Medicine
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity at dopamine receptor D2 on Sf9 cells by [125I]-IABN displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Wake Forest University School of Medicine
Curated by ChEMBL
Wake Forest University School of Medicine
Curated by ChEMBL
Affinity DataKi: 1.04E+4nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to Sigma opioid receptor of guiena pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Wake Forest University School of Medicine
Curated by ChEMBL
Wake Forest University School of Medicine
Curated by ChEMBL
Affinity DataKi: 1.29E+4nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to Sigma opioid receptor of guiena pig brain membraneMore data for this Ligand-Target Pair