Found 96 hits of Enzyme Inhibition Constant Data
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 7.30nMAssay Description:Binding affinity at human histamine H3 receptorMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 7.80nMAssay Description:Binding affinity at rat SERTMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 8.30nMAssay Description:Binding affinity at human histamine H3 receptorMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 8.30nMAssay Description:Binding affinity at rat SERTMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 8.30nMAssay Description:Binding affinity at human histamine H3 receptorMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 8.60nMAssay Description:Binding affinity at human SERTMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 9.30nMAssay Description:Binding affinity at human histamine H3 receptorMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 9.70nMAssay Description:Binding affinity at human histamine H3 receptorMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity at human histamine H3 receptorMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity at human histamine H3 receptorMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity at human histamine H3 receptorMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Binding affinity at human SERTMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Binding affinity at human histamine H3 receptorMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Binding affinity at human histamine H3 receptorMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Binding affinity at human SERTMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Binding affinity at human SERTMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Binding affinity at rat SERTMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Binding affinity at human SERTMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Binding affinity at rat SERTMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Binding affinity at rat SERTMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Binding affinity at human histamine H3 receptorMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Binding affinity at human SERTMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Binding affinity at rat SERTMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Binding affinity at human SERTMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Binding affinity at rat SERTMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Binding affinity at human SERTMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Binding affinity at human histamine H3 receptorMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Binding affinity at human SERTMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Binding affinity at rat SERTMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Binding affinity at human SERTMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Inhibition of [3H]WIN uptake in human DAT expressed in CHO cellsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Binding affinity at rat SERTMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:Binding affinity at human histamine H3 receptorMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 34nMAssay Description:Binding affinity at human SERTMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 36nMAssay Description:Binding affinity at rat SERTMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Binding affinity at human histamine H3 receptorMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Inhibition of [3H]WIN uptake in human DAT expressed in CHO cellsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Binding affinity at human SERTMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 102nMAssay Description:Inhibition of [3H]WIN uptake in human DAT expressed in CHO cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 106nMAssay Description:Inhibition of [3H]nisoxetine uptake in human NET expressed in MDCK cellsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 107nMAssay Description:Binding affinity at human SERTMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 118nMAssay Description:Inhibition of [3H]nisoxetine uptake in human NET expressed in MDCK cellsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Binding affinity at rat SERTMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 121nMAssay Description:Inhibition of [3H]nisoxetine uptake in human NET expressed in MDCK cellsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 135nMAssay Description:Binding affinity at human SERTMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research and Development L.L.C.
Curated by ChEMBL
Affinity DataKi: 7.30E+3nMAssay Description:Binding affinity at human histamine H3 receptorMore data for this Ligand-Target Pair
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