Compile Data Set for Download or QSAR

Found 62 hits of Enzyme Inhibition Constant Data   

TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50478199(CHEMBL410264)copy SMILEScopy InChI
Affinity DataKi:  490nMAssay Description:Displacement of [3]ZM241385 from human adenosine A2A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1NC4PubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University of Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50478203(CHEMBL263372)copy SMILEScopy InChI
Affinity DataKi:  501nMAssay Description:Displacement of [3]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1NC4PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50478212(CHEMBL259430)copy SMILEScopy InChI
Affinity DataKi:  537nMAssay Description:Displacement of [3]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1NC4PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50478212(CHEMBL259430)copy SMILEScopy InChI
Affinity DataKi:  575nMAssay Description:Displacement of [3]ZM241385 from human adenosine A2A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1NC4PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50478196(CHEMBL262351)copy SMILEScopy InChI
Affinity DataKi:  575nMAssay Description:Displacement of [3]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1NC4PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University of Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50478212(CHEMBL259430)copy SMILEScopy InChI
Affinity DataKi:  676nMAssay Description:Displacement of [3]NECA from human adenosine A3 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1NC4PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University of Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50478205(CHEMBL264138)copy SMILEScopy InChI
Affinity DataKi:  1.55E+3nMAssay Description:Displacement of [3]NECA from human adenosine A3 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1NC4PubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University of Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50478199(CHEMBL410264)copy SMILEScopy InChI
Affinity DataKi:  1.74E+3nMAssay Description:Displacement of [3]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1NC4PubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University of Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50478211(CHEMBL262353)copy SMILEScopy InChI
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [3]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1NC4PubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University of Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50478209(CHEMBL263370)copy SMILEScopy InChI
Affinity DataKi:  2.51E+3nMAssay Description:Displacement of [3]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1NC4PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50478197(CHEMBL258849)copy SMILEScopy InChI
Affinity DataKi:  3.09E+3nMAssay Description:Displacement of [3]ZM241385 from human adenosine A2A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1NC4PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50478214(CHEMBL265705)copy SMILEScopy InChI
Affinity DataKi:  3.72E+3nMAssay Description:Displacement of [3]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1NC4PubMed
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