Found 102 hits of Enzyme Inhibition Constant Data
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 1.82E+3nMAssay Description:Inhibition of SYK (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 1.83E+3nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 2.03E+3nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 2.15E+3nMAssay Description:Inhibition of ZAP70 (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 2.23E+3nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >2.27E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 2.45E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >2.50E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >2.50E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >2.50E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >2.50E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 2.98E+3nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >3.33E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: >3.33E+3nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >3.33E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: >3.33E+3nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 3.50E+3nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 3.50E+3nMAssay Description:Inhibition of ZAP70 (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 3.50E+3nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 3.50E+3nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 3.70E+3nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 4.00E+3nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of SYK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of SYK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of SYK (unknown origin)-mediated FCepsilonRI signaling activity by mast cell degranulation assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of SYK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of SYK (unknown origin)-mediated FCepsilonRI signaling activity by mast cell degranulation assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of SYK (unknown origin)-mediated FCepsilonRI signaling activity by mast cell degranulation assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of SYK (unknown origin)-mediated FCepsilonRI signaling activity by mast cell degranulation assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of SYK (unknown origin)-mediated FCepsilonRI signaling activity by mast cell degranulation assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of SYK (unknown origin)-mediated FCepsilonRI signaling activity by mast cell degranulation assayMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
In DepthDetails
Article
BindingDB Entry DOI: 10.7270/Q25Q4VZTPubMedDrugBank
MMDB
PDB
3D Structure (crystal)
BindingDB Entry DOI: 10.7270/Q25Q4VZTPubMedDrugBank
MMDB
PDB
3D Structure (crystal)
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of SYK (unknown origin)-mediated FCepsilonRI signaling activity by mast cell degranulation assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of SYK (unknown origin)-mediated FCepsilonRI signaling activity by mast cell degranulation assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of SYK (unknown origin)-mediated FCepsilonRI signaling activity by mast cell degranulation assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of SYK (unknown origin)-mediated FCepsilonRI signaling activity by mast cell degranulation assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of SYK (unknown origin)-mediated FCepsilonRI signaling activity by mast cell degranulation assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of SYK (unknown origin)-mediated FCepsilonRI signaling activity by mast cell degranulation assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of SYK (unknown origin)-mediated FCepsilonRI signaling activity by mast cell degranulation assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of SYK (unknown origin)-mediated FCepsilonRI signaling activity by mast cell degranulation assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Inhibition of SYK (unknown origin)-mediated FCepsilonRI signaling activity by mast cell degranulation assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 490nMAssay Description:Inhibition of SYK (unknown origin)-mediated FCepsilonRI signaling activity by mast cell degranulation assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Vertex Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 550nMAssay Description:Inhibition of SYK (unknown origin)-mediated FCepsilonRI signaling activity by mast cell degranulation assayMore data for this Ligand-Target Pair