Found 2521 hits of Enzyme Inhibition Constant Data
TargetSerine/threonine-protein kinase SIK3 [59-1321](Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 3.30E+3nMAssay Description:Binding affinity to PAK3More data for this Ligand-Target Pair
Affinity DataKd: 290nMAssay Description:Binding affinity to PIK4CBMore data for this Ligand-Target Pair
Affinity DataKd: 2.10E+3nMAssay Description:Binding affinity to PAK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TNNI3K(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 2.10E+3nMAssay Description:Binding affinity to TNNI3KMore data for this Ligand-Target Pair
Affinity DataKd: 3.70nMAssay Description:Binding affinity to ARK5More data for this Ligand-Target Pair
Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 25nMAssay Description:Binding affinity to AMPK-alpha1More data for this Ligand-Target Pair
Affinity DataKd: 1.20E+3nMAssay Description:Binding affinity to TECMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to DAPK1More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-phosphate 5-kinase type-1 alpha(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 36nMAssay Description:Binding affinity to PIP5K1AMore data for this Ligand-Target Pair
Affinity DataKd: 1.80E+3nMAssay Description:Binding affinity to INSRRMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 110nMAssay Description:Binding affinity to TLK1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MRCK gamma(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to DMPK2More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to RPS6KA6(Kin.Dom.2-C-terminal)More data for this Ligand-Target Pair
TargetEpithelial discoidin domain-containing receptor 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 510nMAssay Description:Binding affinity to DDR1More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 4(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to MAP3K4More data for this Ligand-Target Pair
Affinity DataKd: 27nMAssay Description:Binding affinity to PCTK1More data for this Ligand-Target Pair
Affinity DataKd: 1.20E+3nMAssay Description:Binding affinity to EPHA6More data for this Ligand-Target Pair
Affinity DataKd: 430nMAssay Description:Binding affinity to LCKMore data for this Ligand-Target Pair
Affinity DataKd: 530nMAssay Description:Binding affinity to CDK9More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 2.50E+3nMAssay Description:Binding affinity to MAP4K2More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to PAK6More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to ULK1More data for this Ligand-Target Pair
Affinity DataKd: 140nMAssay Description:Binding affinity to PRKCHMore data for this Ligand-Target Pair
Affinity DataKd: 370nMAssay Description:Binding affinity to PRKG1More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to NEK5More data for this Ligand-Target Pair
Affinity DataKd: 220nMAssay Description:Binding affinity to PLK1More data for this Ligand-Target Pair
Affinity DataKd: 380nMAssay Description:Binding affinity to PRKD2More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to BRSK1More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to PIK3CDMore data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to TYK2(JH2domain-pseudokinase)More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to MST3More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to EPHB2More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 330nMAssay Description:Binding affinity to DYRK1BMore data for this Ligand-Target Pair
Affinity DataKd: 960nMAssay Description:Binding affinity to AAK1More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 4(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to MAP3K4More data for this Ligand-Target Pair
Affinity DataKd: 1.70E+3nMAssay Description:Binding affinity to FGFR3More data for this Ligand-Target Pair
Affinity DataKd: 8.10nMAssay Description:Binding affinity to PRKD2More data for this Ligand-Target Pair
TargetTestis-specific serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 4.80E+3nMAssay Description:Binding affinity to TSSK1BMore data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 6.20E+3nMAssay Description:Binding affinity to AKT3More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to TAOK1More data for this Ligand-Target Pair
TargetMacrophage-stimulating protein receptor(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to MST1RMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit beta(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CAMK2BMore data for this Ligand-Target Pair
Affinity DataKd: 1nMAssay Description:Binding affinity to DRAK1More data for this Ligand-Target Pair
Affinity DataKd: 270nMAssay Description:Binding affinity to ALKMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to INSRMore data for this Ligand-Target Pair
Affinity DataKd: 840nMAssay Description:Binding affinity to DLKMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to TAO1More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 640nMAssay Description:Binding affinity to SRCMore data for this Ligand-Target Pair
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