Found 176 hits of Enzyme Inhibition Constant Data
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human adrenergic beta-1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human 5-HT7 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human NK2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human D2S agonist site receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human adenosine A3 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to Lyn by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human histamine H2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human muscarinic M1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human muscarinic M3 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human adenosine A1 receptor agonist site by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human 5HT2C receptor agonist site by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to 5-HT1B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human adenosine A3 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human 5-HT2B agonist site receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to kappa opioid receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human glucocorticoid receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human UT1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to 5-HT1B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
H. Lundbeck A/S
Curated by ChEMBL
H. Lundbeck A/S
Curated by ChEMBL
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human NE transporter by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human NK2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human ETA receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to adrenergic alpha2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to Lyn by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human dopamine D1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human histamine H2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human histamine H3 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
H. Lundbeck A/S
Curated by ChEMBL
H. Lundbeck A/S
Curated by ChEMBL
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to nAChR alpha4beta2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human CCK2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human NK1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to adrenergic beta2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human adenosine A2A receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
H. Lundbeck A/S
Curated by ChEMBL
H. Lundbeck A/S
Curated by ChEMBL
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to ML2 (MT3) receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human CB1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to adrenergic beta2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human neuropeptide Y1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human 5-HT2B agonist site receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human CB1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human adenosine A1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human muscarinic M4 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
H. Lundbeck A/S
Curated by ChEMBL
H. Lundbeck A/S
Curated by ChEMBL
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to nAChR alpha4beta2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to MAOA by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human dopamine D2S receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human muscarinic M4 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human dopamine transporter by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human 5-HT3 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human mu opioid receptor agonist site by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human adrenergic Alpha-1D receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human neuropeptide Y1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to I1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human acetylcholine esterase by radioligand displacement assayMore data for this Ligand-Target Pair
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