Found 81 hits of Enzyme Inhibition Constant Data
Affinity DataIC50: 18nMAssay Description:Inhibition of ALK enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of ALK Tyr1604 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibition of ALK enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:Inhibition of ALK Tyr1604 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Inhibition of ALK Tyr1604 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Inhibition of ALK Tyr1604 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 109nMAssay Description:Inhibition of ALK Tyr1604 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 144nMAssay Description:Inhibition of ALK Tyr1604 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 147nMAssay Description:Inhibition of ALK Tyr1604 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 231nMAssay Description:Inhibition of INSR expressed in CHO cells assessed as inhibition of receptor phosphorylation pre-incubated before insulin stimulation by Meso-Scale D...More data for this Ligand-Target Pair
Affinity DataIC50: 345nMAssay Description:Inhibition of ALK Tyr1604 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 536nMAssay Description:Inhibition of INSR expressed in CHO cells assessed as inhibition of receptor phosphorylation pre-incubated before insulin stimulation by Meso-Scale D...More data for this Ligand-Target Pair
Affinity DataIC50: 562nMAssay Description:Inhibition of ALK Tyr1604 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.12E+3nMAssay Description:Inhibition of c-Met enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 5.92E+3nMAssay Description:Inhibition of c-Met enzymeMore data for this Ligand-Target Pair
Affinity DataKd: 8.20nMAssay Description:Binding affinity to human LTK by Ambit titration assayMore data for this Ligand-Target Pair
Affinity DataKd: 72nMAssay Description:Binding affinity to human MER by Ambit titration assayMore data for this Ligand-Target Pair
Affinity DataKd: 28nMAssay Description:Binding affinity to human LCK by Ambit titration assayMore data for this Ligand-Target Pair
Affinity DataKd: 2.5nMAssay Description:Binding affinity to human LTK by Ambit titration assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.60E+3nMAssay Description:Binding affinity to human AXL by Ambit titration assayMore data for this Ligand-Target Pair
Affinity DataKd: 5.60nMAssay Description:Binding affinity to human IRAK1 by Ambit titration assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Amgen Inc.
Curated by ChEMBL
Amgen Inc.
Curated by ChEMBL
Affinity DataKd: 11nMAssay Description:Binding affinity to human MAP4K2 by Ambit titration assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Amgen Inc.
Curated by ChEMBL
Amgen Inc.
Curated by ChEMBL
Affinity DataKd: 25nMAssay Description:Binding affinity to human MAP4K2 by Ambit titration assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.360nMAssay Description:Binding affinity to human ALK by Ambit titration assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.240nMAssay Description:Binding affinity to human ALK by Ambit titration assayMore data for this Ligand-Target Pair
Affinity DataKd: 18nMAssay Description:Binding affinity to human MER by Ambit titration assayMore data for this Ligand-Target Pair
Affinity DataKd: 42nMAssay Description:Binding affinity to human FLT3 by Ambit titration assayMore data for this Ligand-Target Pair
Affinity DataKd: 72nMAssay Description:Binding affinity to human INSR by Ambit titration assayMore data for this Ligand-Target Pair
Affinity DataKd: 110nMAssay Description:Binding affinity to human LCK by Ambit titration assayMore data for this Ligand-Target Pair
Affinity DataKd: 5.70nMAssay Description:Binding affinity to human IRAK1 by Ambit titration assayMore data for this Ligand-Target Pair
Affinity DataKd: 29nMAssay Description:Binding affinity to human AXL by Ambit titration assayMore data for this Ligand-Target Pair