Compile Data Set for Download or QSAR

Found 154 hits of Enzyme Inhibition Constant Data   

TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431349(CHEMBL2348648)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Inhibition of human recombinant His6 tagged CDK2/Cyclin A expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431354(CHEMBL2348643)copy SMILEScopy InChI
Affinity DataKi:  22nMAssay Description:Inhibition of human recombinant His6 tagged CDK9/CyclinT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431350(CHEMBL2348647)copy SMILEScopy InChI
Affinity DataKi:  24nMAssay Description:Inhibition of human recombinant His6 tagged CDK1/Cyclin B expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431354(CHEMBL2348643)copy SMILEScopy InChI
Affinity DataKi:  26nMAssay Description:Inhibition of human recombinant His6 tagged CDK2/Cyclin A expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431351(CHEMBL2348646)copy SMILEScopy InChI
Affinity DataKi:  26nMAssay Description:Inhibition of human recombinant His6 tagged CDK1/Cyclin B expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431358(CHEMBL2348638)copy SMILEScopy InChI
Affinity DataKi:  34nMAssay Description:Inhibition of human recombinant His6 tagged CDK2/Cyclin A expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431352(CHEMBL2348645)copy SMILEScopy InChI
Affinity DataKi:  35nMAssay Description:Inhibition of human recombinant His6 tagged CDK1/Cyclin B expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431353(CHEMBL2348644)copy SMILEScopy InChI
Affinity DataKi:  39nMAssay Description:Inhibition of human recombinant His6 tagged CDK2/Cyclin A expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431337(CHEMBL2348845)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431355(CHEMBL2348642)copy SMILEScopy InChI
Affinity DataKi:  42nMAssay Description:Inhibition of human recombinant His6 tagged CDK1/Cyclin B expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431351(CHEMBL2348646)copy SMILEScopy InChI
Affinity DataKi:  42nMAssay Description:Inhibition of human recombinant His6 tagged CDK2/Cyclin A expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431352(CHEMBL2348645)copy SMILEScopy InChI
Affinity DataKi:  42nMAssay Description:Inhibition of human recombinant His6 tagged CDK2/Cyclin A expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431356(CHEMBL2348641)copy SMILEScopy InChI
Affinity DataKi:  43nMAssay Description:Inhibition of human recombinant His6 tagged CDK1/Cyclin B expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431356(CHEMBL2348641)copy SMILEScopy InChI
Affinity DataKi:  43nMAssay Description:Inhibition of human recombinant His6 tagged CDK2/Cyclin A expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431348(CHEMBL2348649)copy SMILEScopy InChI
Affinity DataKi:  45nMAssay Description:Inhibition of human recombinant His6 tagged CDK2/Cyclin A expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431354(CHEMBL2348643)copy SMILEScopy InChI
Affinity DataKi:  45nMAssay Description:Inhibition of human recombinant His6 tagged CDK1/Cyclin B expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431347(CHEMBL2348650)copy SMILEScopy InChI
Affinity DataKi:  47nMAssay Description:Inhibition of human recombinant His6 tagged CDK1/Cyclin B expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431340(CHEMBL2348842)copy SMILEScopy InChI
Affinity DataKi:  47nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431338(CHEMBL2348844)copy SMILEScopy InChI
Affinity DataKi:  54nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431355(CHEMBL2348642)copy SMILEScopy InChI
Affinity DataKi:  56nMAssay Description:Inhibition of human recombinant His6 tagged CDK2/Cyclin A expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431358(CHEMBL2348638)copy SMILEScopy InChI
Affinity DataKi:  62nMAssay Description:Inhibition of human recombinant His6 tagged CDK1/Cyclin B expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431339(CHEMBL2348843)copy SMILEScopy InChI
Affinity DataKi:  64nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431334(CHEMBL2348848)copy SMILEScopy InChI
Affinity DataKi:  66nMAssay Description:Inhibition of human recombinant His6 tagged CDK9/CyclinT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431355(CHEMBL2348642)copy SMILEScopy InChI
Affinity DataKi:  68nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431353(CHEMBL2348644)copy SMILEScopy InChI
Affinity DataKi:  71nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431353(CHEMBL2348644)copy SMILEScopy InChI
Affinity DataKi:  79nMAssay Description:Inhibition of human recombinant His6 tagged CDK1/Cyclin B expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431347(CHEMBL2348650)copy SMILEScopy InChI
Affinity DataKi:  85nMAssay Description:Inhibition of human recombinant His6 tagged CDK2/Cyclin A expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431348(CHEMBL2348649)copy SMILEScopy InChI
Affinity DataKi:  88nMAssay Description:Inhibition of human recombinant His6 tagged CDK1/Cyclin B expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431360(CHEMBL2347597)copy SMILEScopy InChI
Affinity DataKi:  91nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431346(CHEMBL2348651)copy SMILEScopy InChI
Affinity DataKi:  91nMAssay Description:Inhibition of human recombinant His6 tagged CDK1/Cyclin B expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431356(CHEMBL2348641)copy SMILEScopy InChI
Affinity DataKi:  92nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431357(CHEMBL2348639)copy SMILEScopy InChI
Affinity DataKi:  98nMAssay Description:Inhibition of human recombinant His6 tagged CDK9/CyclinT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431347(CHEMBL2348650)copy SMILEScopy InChI
Affinity DataKi:  111nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50425010(CHEMBL2312183)copy SMILEScopy InChI
Affinity DataKi:  114nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431346(CHEMBL2348651)copy SMILEScopy InChI
Affinity DataKi:  131nMAssay Description:Inhibition of human recombinant His6 tagged CDK2/Cyclin A expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431344(CHEMBL2348653)copy SMILEScopy InChI
Affinity DataKi:  134nMAssay Description:Inhibition of human recombinant His6 tagged CDK9/CyclinT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431341(CHEMBL2348841)copy SMILEScopy InChI
Affinity DataKi:  154nMAssay Description:Inhibition of human recombinant His6 tagged CDK1/Cyclin B expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431348(CHEMBL2348649)copy SMILEScopy InChI
Affinity DataKi:  155nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431341(CHEMBL2348841)copy SMILEScopy InChI
Affinity DataKi:  156nMAssay Description:Inhibition of human recombinant His6 tagged CDK9/CyclinT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431334(CHEMBL2348848)copy SMILEScopy InChI
Affinity DataKi:  176nMAssay Description:Inhibition of human recombinant His6 tagged CDK1/Cyclin B expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431350(CHEMBL2348647)copy SMILEScopy InChI
Affinity DataKi:  193nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431345(CHEMBL2348652)copy SMILEScopy InChI
Affinity DataKi:  195nMAssay Description:Inhibition of human recombinant His6 tagged CDK1/Cyclin B expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431346(CHEMBL2348651)copy SMILEScopy InChI
Affinity DataKi:  210nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431341(CHEMBL2348841)copy SMILEScopy InChI
Affinity DataKi:  226nMAssay Description:Inhibition of human recombinant His6 tagged CDK2/Cyclin A expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431343(CHEMBL2348654)copy SMILEScopy InChI
Affinity DataKi:  245nMAssay Description:Inhibition of human recombinant His6 tagged CDK9/CyclinT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431335(CHEMBL2348847)copy SMILEScopy InChI
Affinity DataKi:  255nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50425011(CHEMBL2312182)copy SMILEScopy InChI
Affinity DataKi:  260nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431336(CHEMBL2348846)copy SMILEScopy InChI
Affinity DataKi:  273nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431342(CHEMBL2348840)copy SMILEScopy InChI
Affinity DataKi:  278nMAssay Description:Inhibition of human recombinant His6 tagged CDK9/CyclinT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431343(CHEMBL2348654)copy SMILEScopy InChI
Affinity DataKi:  282nMAssay Description:Inhibition of human recombinant His6 tagged CDK2/Cyclin A expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
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