Found 100 hits of Enzyme Inhibition Constant Data
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of TAK1 in human HCT116 cells assessed as inhibition of TNF-alpha-stimulated JNK phosphorylationMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of TAK1 in human HCT116 cells assessed as inhibition of TNF-alpha-stimulated JNK phosphorylationMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of TAK1 in human HCT116 cells assessed as inhibition of TNF-alpha-stimulated JNK phosphorylationMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of TAK1 in human HCT116 cells assessed as inhibition of TNF-alpha-stimulated JNK phosphorylationMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of TAK1 in human HCT116 cells assessed as inhibition of TNF-alpha-stimulated JNK phosphorylationMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of TAK1 in human HCT116 cells assessed as inhibition of TNF-alpha-stimulated JNK phosphorylationMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of TAK1 in human HCT116 cells assessed as inhibition of TNF-alpha-stimulated JNK phosphorylationMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of TAK1 in human HCT116 cells assessed as inhibition of TNF-alpha-stimulated JNK phosphorylationMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of TAK1 in human HCT116 cells assessed as inhibition of TNF-alpha-stimulated JNK phosphorylationMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of TAK1 in human HCT116 cells assessed as inhibition of TNF-alpha-stimulated JNK phosphorylationMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of TAK1 in human HCT116 cells assessed as inhibition of TNF-alpha-stimulated JNK phosphorylationMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of TAK1 in human HCT116 cells assessed as inhibition of TNF-alpha-stimulated JNK phosphorylationMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of TAK1 in human HCT116 cells assessed as inhibition of TNF-alpha-stimulated JNK phosphorylationMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of TAK1 in human HCT116 cells assessed as inhibition of TNF-alpha-stimulated JNK phosphorylationMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of TAK1 in human HCT116 cells assessed as inhibition of TNF-alpha-stimulated JNK phosphorylationMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of TAK1 in human HCT116 cells assessed as inhibition of TNF-alpha-stimulated JNK phosphorylationMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of TAK1 in human HCT116 cells assessed as inhibition of TNF-alpha-stimulated JNK phosphorylationMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of TAK1 in human HCT116 cells assessed as inhibition of TNF-alpha-stimulated JNK phosphorylationMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 1.75E+4nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of TAK1 in human HCT116 cells assessed as inhibition of TNF-alpha-stimulated JNK phosphorylationMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 2.57E+4nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1(Homo sapiens (Human))
OSI Pharmaceuticals LLC
Curated by ChEMBL
OSI Pharmaceuticals LLC
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair