Compile Data Set for Download or QSAR

Found 304 hits of Enzyme Inhibition Constant Data   

TargetVitamin K-dependent protein C(Homo sapiens (Human))
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50532400(CHEMBL4549153)copy SMILEScopy InChI
Affinity DataKi:  2.12E+5nMAssay Description:Inhibition of human activated Protein C using Mes-DArg-Pro-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377D5TPubMed
TargetVitamin K-dependent protein C(Homo sapiens (Human))
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50532400(CHEMBL4549153)copy SMILEScopy InChI
Affinity DataKi:  2.12E+5nMAssay Description:Inhibition of human activated Protein C using Mes-DArg-Pro-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377D5TPubMed
TargetCoagulation factor X(Homo sapiens (Human))
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50532395(CHEMBL4547050)copy SMILEScopy InChI
Affinity DataKi:  4.05E+5nMAssay Description:Inhibition of human f10a using Mes-DArg-Pro-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377D5TPubMed
TargetCoagulation factor X(Homo sapiens (Human))
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50532395(CHEMBL4547050)copy SMILEScopy InChI
Affinity DataKi:  4.05E+5nMAssay Description:Inhibition of human f10a using Mes-DArg-Pro-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377D5TPubMed
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