Found 260 hits of Enzyme Inhibition Constant Data
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of human ALDH1A1 using all-trans-retinal as substrate preincubated for 15 mins followed by substrate addition measured for 30 mins by fluo...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of ALDH1A1 in human MIAPaCa2 cells after 30 mins by aldefluor assayMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of ALDH1A1 in human MIAPaCa2 cells after 30 mins by aldefluor assayMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of ALDH1A1 in human MIAPaCa2 cells after 30 mins by aldefluor assayMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of ALDH1A1 in human SKOV3TR cells assessed as potentiation of paclitaxel-mediated cytotoxicity by measuring paclitaxel IC50 at 10 uM after...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of ALDH1A1 in human MIAPaCa2 cells after 30 mins by aldefluor assayMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of ALDH1A1 in human MIAPaCa2 cells after 30 mins by aldefluor assayMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of ALDH1A1 in human MIAPaCa2 cells after 30 mins by aldefluor assayMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of ALDH1A1 in human SKOV3TR cells assessed as potentiation of paclitaxel-mediated cytotoxicity by measuring paclitaxel IC50 at 30 uM after...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of ALDH1A1 in human MIAPaCa2 cells after 30 mins by aldefluor assayMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of ALDH1A1 in human MIAPaCa2 cells after 30 mins by aldefluor assayMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of ALDH1A1 in human MIAPaCa2 cells after 30 mins by aldefluor assayMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of ALDH1A1 in human MIAPaCa2 cells after 30 mins by aldefluor assayMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibition of ALDH1A1 in human MIAPaCa2 cells after 30 mins by aldefluor assayMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of ALDH1A1 in human MIAPaCa2 cells after 30 mins by aldefluor assayMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of ALDH1A1 in human MIAPaCa2 cells after 30 mins by aldefluor assayMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of ALDH1A1 in human MIAPaCa2 cells after 30 mins by aldefluor assayMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of ALDH1A1 in human MIAPaCa2 cells after 30 mins by aldefluor assayMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of ALDH1A1 in human MIAPaCa2 cells after 30 mins by aldefluor assayMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of ALDH1A1 in human MIAPaCa2 cells after 30 mins by aldefluor assayMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Inhibition of ALDH1A1 in human MIAPaCa2 cells after 30 mins by aldefluor assayMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:Inhibition of human ALDH1A1 using all-trans-retinal as substrate preincubated for 15 mins followed by substrate addition measured for 30 mins by fluo...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human ALDH1A1 using NAD+/propionaldehyde as substrate/cofactor preincubated for 15 mins followed by substrate/cofactor addition measure...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase 1A1(Homo sapiens (Human))
National Center for Advancing Translational Sciences
Curated by ChEMBL
National Center for Advancing Translational Sciences
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Inhibition of ALDH1A1 in human MIAPaCa2 cells after 30 mins by aldefluor assayMore data for this Ligand-Target Pair