Found 51 hits of Enzyme Inhibition Constant Data
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 61nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues) using biotin-labelled H3K4me2 (1 to 24 residues) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 66nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues) using biotin-labelled H3K4me2 (1 to 24 residues) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 84nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues) using biotin-labelled H3K4me2 (1 to 24 residues) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 109nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues) using biotin-labelled H3K4me2 (1 to 24 residues) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 124nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues) using biotin-labelled H3K4me2 (1 to 24 residues) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 146nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues) using biotin-labelled H3K4me2 (1 to 24 residues) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 184nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues) using biotin-labelled H3K4me2 (1 to 24 residues) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 187nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues) using biotin-labelled H3K4me2 (1 to 24 residues) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 211nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues) using biotin-labelled H3K4me2 (1 to 24 residues) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 241nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues) using biotin-labelled H3K4me2 (1 to 24 residues) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 242nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues) using biotin-labelled H3K4me2 (1 to 24 residues) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 252nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues) using biotin-labelled H3K4me2 (1 to 24 residues) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 303nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues) using biotin-labelled H3K4me2 (1 to 24 residues) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues) using biotin-labelled H3K4me2 (1 to 24 residues) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Inhibition of MAOB (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 692nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues) using biotin-labelled H3K4me2 (1 to 24 residues) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of MAOA (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 1.16E+3nMAssay Description:Inhibition of MAOB (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues) using biotin-labelled H3K4me2 (1 to 24 residues) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of MAOB (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 2.23E+3nMAssay Description:Inhibition of MAOA (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of MAOA (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 4.55E+3nMAssay Description:Inhibition of MAOA (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 4.81E+3nMAssay Description:Inhibition of MAOB (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 6.05E+3nMAssay Description:Inhibition of MAOB (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 8.27E+3nMAssay Description:Inhibition of MAOA (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 8.57E+3nMAssay Description:Inhibition of MAOA (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 9.19E+3nMAssay Description:Inhibition of MAOA (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 9.63E+3nMAssay Description:Inhibition of MAOB (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of MAOA (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 1.29E+4nMAssay Description:Inhibition of MAOA (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 2.04E+4nMAssay Description:Inhibition of MAOB (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 2.08E+4nMAssay Description:Inhibition of MAOA (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of MAOA (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 2.19E+4nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues) using biotin-labelled H3K4me2 (1 to 24 residues) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of MAOB (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 2.88E+4nMAssay Description:Inhibition of MAOB (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 3.67E+4nMAssay Description:Inhibition of MAOB (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 4.03E+4nMAssay Description:Inhibition of MAOB (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 4.09E+4nMAssay Description:Inhibition of MAOA (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 4.75E+4nMAssay Description:Inhibition of MAOA (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 4.95E+4nMAssay Description:Inhibition of MAOB (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 5.64E+4nMAssay Description:Inhibition of MAOA (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 6.59E+4nMAssay Description:Inhibition of MAOA (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 7.16E+4nMAssay Description:Inhibition of MAOB (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 7.56E+4nMAssay Description:Inhibition of MAOB (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 9.56E+4nMAssay Description:Inhibition of MAOB (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of MAOA (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of MAOA (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Liaoning Shihua University
Curated by ChEMBL
Liaoning Shihua University
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of MAOB (unknown origin) by Promega MAO-Glo assayMore data for this Ligand-Target Pair