Found 86 hits of Enzyme Inhibition Constant Data
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 9.5nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 38nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 79nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 79nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 86nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 95nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 167nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 178nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 201nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 203nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 207nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 212nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 215nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 328nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 354nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 383nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 537nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 725nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 739nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 749nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 763nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 868nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 3.35E+3nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: >4.72E+3nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: >5.71E+3nMAssay Description:Displacement of [125I]BTX from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 1.65nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 15.6nMAssay Description:Displacement of [3H]epibatidine from alpha3 nAChR in human IMR32 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 1.04E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 1.07E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 1.39E+3nMAssay Description:Displacement of [3H]epibatidine from alpha3 nAChR in human IMR32 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 1.78E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 2.04E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 2.09E+3nMAssay Description:Displacement of [3H]epibatidine from alpha3 nAChR in human IMR32 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 2.62E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 3.16E+3nMAssay Description:Displacement of [3H]LY278584 from human 5HT3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair