Found 7 hits of Enzyme Inhibition Constant Data
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Washington University in Saint Louis
Curated by ChEMBL
Washington University in Saint Louis
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:Inhibition of PARP-1 (unknown origin) assessed as NAD+ consumption after 20 mins by fluorometric analysis in presence of activated DNAMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Washington University in Saint Louis
Curated by ChEMBL
Washington University in Saint Louis
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of PARP-1 (unknown origin) assessed as NAD+ consumption after 20 mins by fluorometric analysis in presence of activated DNAMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Washington University in Saint Louis
Curated by ChEMBL
Washington University in Saint Louis
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of PARP-1 (unknown origin) assessed as NAD+ consumption after 20 mins by fluorometric analysis in presence of activated DNAMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Washington University in Saint Louis
Curated by ChEMBL
Washington University in Saint Louis
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of PARP-1 (unknown origin) assessed as NAD+ consumption after 20 mins by fluorometric analysis in presence of activated DNAMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Washington University in Saint Louis
Curated by ChEMBL
Washington University in Saint Louis
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of PARP-1 (unknown origin) assessed as NAD+ consumption after 20 mins by fluorometric analysis in presence of activated DNAMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Washington University in Saint Louis
Curated by ChEMBL
Washington University in Saint Louis
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of PARP-1 (unknown origin) assessed as NAD+ consumption after 20 mins by fluorometric analysis in presence of activated DNAMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Washington University in Saint Louis
Curated by ChEMBL
Washington University in Saint Louis
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of PARP-1 (unknown origin) assessed as NAD+ consumption after 20 mins by fluorometric analysis in presence of activated DNAMore data for this Ligand-Target Pair