Compile Data Set for Download or QSAR

Found 13 hits of Enzyme Inhibition Constant Data   

TargetAdenosine receptor A3(Homo sapiens (Human))
Panjab University

Curated by ChEMBL
LigandPNGBDBM50496138(CHEMBL3121727)copy SMILEScopy InChI
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-HEMADO from human recombinant adenosine A3 receptor expressed in CHO cell membranes after 3 hrs by microbeta counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9SC2PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Panjab University

Curated by ChEMBL
LigandPNGBDBM50496137(CHEMBL3121723)copy SMILEScopy InChI
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]-HEMADO from human recombinant adenosine A3 receptor expressed in CHO cell membranes after 3 hrs by microbeta counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9SC2PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Panjab University

Curated by ChEMBL
LigandPNGBDBM50496131(CHEMBL3121724)copy SMILEScopy InChI
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]-HEMADO from human recombinant adenosine A3 receptor expressed in CHO cell membranes after 3 hrs by microbeta counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9SC2PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Panjab University

Curated by ChEMBL
LigandPNGBDBM50496136(CHEMBL3121722)copy SMILEScopy InChI
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]-HEMADO from human recombinant adenosine A3 receptor expressed in CHO cell membranes after 3 hrs by microbeta counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9SC2PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Panjab University

Curated by ChEMBL
LigandPNGBDBM50496141(CHEMBL3121721)copy SMILEScopy InChI
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]-HEMADO from human recombinant adenosine A3 receptor expressed in CHO cell membranes after 3 hrs by microbeta counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9SC2PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Panjab University

Curated by ChEMBL
LigandPNGBDBM50496142(CHEMBL3121728)copy SMILEScopy InChI
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H]-HEMADO from human recombinant adenosine A3 receptor expressed in CHO cell membranes after 3 hrs by microbeta counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9SC2PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Panjab University

Curated by ChEMBL
LigandPNGBDBM50496135(CHEMBL3121720)copy SMILEScopy InChI
Affinity DataKi:  9.40nMAssay Description:Displacement of [3H]-HEMADO from human recombinant adenosine A3 receptor expressed in CHO cell membranes after 3 hrs by microbeta counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9SC2PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Panjab University

Curated by ChEMBL
LigandPNGBDBM50496134(CHEMBL3121726)copy SMILEScopy InChI
Affinity DataKi: >10nMAssay Description:Displacement of [3H]-HEMADO from human recombinant adenosine A3 receptor expressed in CHO cell membranes after 3 hrs by microbeta counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9SC2PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Panjab University

Curated by ChEMBL
LigandPNGBDBM50496132(CHEMBL3121729)copy SMILEScopy InChI
Affinity DataKi: >30nMAssay Description:Displacement of [3H]-HEMADO from human recombinant adenosine A3 receptor expressed in CHO cell membranes after 3 hrs by microbeta counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9SC2PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Panjab University

Curated by ChEMBL
LigandPNGBDBM50496133(CHEMBL3121725)copy SMILEScopy InChI
Affinity DataKi: >30nMAssay Description:Displacement of [3H]-HEMADO from human recombinant adenosine A3 receptor expressed in CHO cell membranes after 3 hrs by microbeta counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9SC2PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Panjab University

Curated by ChEMBL
LigandPNGBDBM50496130(CHEMBL3121731)copy SMILEScopy InChI
Affinity DataKi: >30nMAssay Description:Displacement of [3H]-HEMADO from human recombinant adenosine A3 receptor expressed in CHO cell membranes after 3 hrs by microbeta counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9SC2PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Panjab University

Curated by ChEMBL
LigandPNGBDBM50496139(CHEMBL3121732)copy SMILEScopy InChI
Affinity DataKi: >30nMAssay Description:Displacement of [3H]-HEMADO from human recombinant adenosine A3 receptor expressed in CHO cell membranes after 3 hrs by microbeta counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9SC2PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Panjab University

Curated by ChEMBL
LigandPNGBDBM50496140(CHEMBL3121730)copy SMILEScopy InChI
Affinity DataKi: >30nMAssay Description:Displacement of [3H]-HEMADO from human recombinant adenosine A3 receptor expressed in CHO cell membranes after 3 hrs by microbeta counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9SC2PubMed
Displayed 1 to 50 (of 52 total ) | Next | Last >>* indicates data uncertainty>20%